SCHEMBL23116558

SCHEMBL23116558

CN(C)C[C@H](Cc1ccccc1)NC(=O)c1ccccc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTRB1 P17538 6/20 0.66
HDAC4 P56524 4/20 0.60
HDAC6 Q9UBN7 4/20 0.60
PIN1 Q13526 1/20 0.58
CTSL P07711 3/20 0.57
ROCK2 O75116 1/20 0.51
RPS6KA5 O75582 1/20 0.51
RPS6KA4 O75676 1/20 0.51
PRKACA P17612 1/20 0.51
MAPK1 P28482 1/20 0.51
GSK3A P49840 1/20 0.51
GSK3B P49841 1/20 0.51
IRAK1 P51617 1/20 0.51
PRKX P51817 1/20 0.51
ROCK1 Q13464 1/20 0.51
PRKG1 Q13976 1/20 0.51
PKN2 Q16513 1/20 0.51
CLK4 Q9HAZ1 1/20 0.51
SGK2 Q9HBY8 1/20 0.51
ECE1 P42892 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10952300 1.00 CTRB1 (0.66) CTRB1HDAC4HDAC6PIN1CTSL
SCHEMBL13061025 0.88 CTRB1 (0.52) CTRB1HDAC4HDAC6PIN1CTSL
SCHEMBL13005491 0.87 CTRB1 (0.51) CTRB1HDAC4HDAC6PIN1CTSL
SCHEMBL1570133 0.86 HDAC4 (0.49) CTRB1HDAC4HDAC6MAPK1RAB9A
SCHEMBL21496635 0.86 HDAC4 (0.49) CTRB1HDAC4HDAC6MAPK1RAB9A
SCHEMBL23116580 0.84 CTRB1 (0.54) CTRB1HDAC4HDAC6MAPK1RAB9A
SCHEMBL23116581 0.84 CTRB1 (0.54) CTRB1HDAC4HDAC6MAPK1RAB9A
SCHEMBL13060697 0.84 MME (0.52) CTRB1HDAC4HDAC6CTSLALDH1A1
SCHEMBL8254900 0.83 CTRB1 (0.48) CTRB1HDAC4HDAC6MAPK1RAB9A
SCHEMBL13005665 0.83 MME (0.51) CTRB1HDAC4HDAC6CTSLALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112312902-B Pd (II) -catalyzed enantioselective C-H arylation of free carboxylic acids 斯克里普斯研究学院 2022-02-18 CN disclosed
US-20210087131-A1 PD(II)-CATALYZED ENANTIOSELECTIVE C-H ARYLATION OF FREE CARBOXYLIC ACIDS THE SCRIPPS RESEARCH INSTITUTE 2021-03-25 US disclosed
CN-112312902-A Pd (II) -catalyzed enantioselective C-H arylation of free carboxylic acids 斯克里普斯研究学院 2021-02-02 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210087131-A1 PD(II)-CATALYZED ENANTIOSELECTIVE C-H ARYLATION OF FREE CARBOXYLIC ACIDS PDCD1, PDK3, PDCD1LG2 CTRB1 2266/4885HDAC4 1480/4885HDAC6 847/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.