SCHEMBL23119613

SCHEMBL23119613

COCCOC1CCN(c2ccc(Br)cc2NS(=O)(=O)c2cccc(C(F)(F)F)c2)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.52
ERAP1 Q9NZ08 1/20 0.46
ALDH1A1 P00352 5/20 0.46
LMNA P02545 5/20 0.46
LIPC P11150 1/20 0.45
LIPG Q9Y5X9 1/20 0.45
KDM4E B2RXH2 2/20 0.44
MAPT P10636 2/20 0.44
TDP1 Q9NUW8 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
GAA P10253 1/20 0.44
ALOX15 P16050 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.42
HTR6 P50406 4/20 0.40
DNMT1 P26358 1/20 0.40
CASP6 P55212 1/20 0.40
DRD2 P14416 1/20 0.39
ADRA1D P25100 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23119684 0.83 NPSR1 (0.56) NPSR1ERAP1ALDH1A1LMNAKDM4E
SCHEMBL23119377 0.83 NPSR1 (0.56) NPSR1ERAP1ALDH1A1LMNAKDM4E
SCHEMBL23093745 0.81 RORC (0.51)
SCHEMBL30593065 0.81 RORC (0.51)
SCHEMBL23119482 0.79 LMNA (0.72) NPSR1ERAP1ALDH1A1LMNAKDM4E
SCHEMBL23119610 0.77 NPSR1 (0.55) NPSR1ERAP1ALDH1A1LMNAKDM4E
SCHEMBL23119663 0.77 ERAP1 (0.53) NPSR1ERAP1ALDH1A1LMNAKDM4E
SCHEMBL7568254 0.72 MEN1 (0.57) NPSR1LMNAGAA
SCHEMBL29666321 0.70 MEN1 (0.55) NPSR1ALDH1A1LMNAGAA
SCHEMBL18302531 0.70 MEN1 (0.55) NPSR1ALDH1A1LMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021047407-A1 BIARYL COMPOUND, PHARMACEUTICAL COMPOSITION COMPRISING SAME, PREPARATION METHOD THEREFOR, AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2021-03-18 WO disclosed