SCHEMBL23123776

SCHEMBL23123776

Cn1c(=O)oc2cc(N3CC(C)(C)N(C(=O)O)CC3=O)ccc21

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
HPGD P15428 1/20 0.44
CYP11B2 P19099 1/20 0.40
ASAH1 Q13510 1/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
POLB P06746 2/20 0.38
TP53 P04637 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
PKM P14618 2/20 0.37
TSHR P16473 1/20 0.37
HTR1A P08908 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29709631 0.86 ALDH1A1 (0.37) ALDH1A1HPGDCYP11B2ASAH1KDM4E
SCHEMBL24792962 0.86 ALDH1A1 (0.37) ALDH1A1HPGDCYP11B2ASAH1KDM4E
SCHEMBL23123381 0.81 MEN1 (0.45) ALDH1A1HPGDCYP11B2ASAH1KDM4E
SCHEMBL23123109 0.81 ASAH1 (0.64) ASAH1
SCHEMBL23122327 0.79 ALDH1A1 (0.44) ALDH1A1HPGDCYP11B2ASAH1KDM4E
SCHEMBL23123472 0.78 ASAH1 (0.47) ALDH1A1HPGDCYP11B2ASAH1KDM4E
SCHEMBL23122239 0.78 NOS1 (0.40) ALDH1A1KDM4EMEN1KMT2ATDP1
SCHEMBL24793637 0.77 PKM (0.43) ALDH1A1HPGDCYP11B2KDM4EMEN1
Hydrochloric Acid SCHEMBL23123134 0.76 PKM (0.42) ALDH1A1HPGDCYP11B2KDM4EMEN1
SCHEMBL23123105 0.75 KDM4E (0.37) ALDH1A1HPGDKDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021055627-A1 SUBSTITUTED N-HETEROCYCLIC CARBOXAMIDES AS ACID CERAMIDASE INHIBITORS AND THEIR USE AS MEDICAMENTS BIAL- BIOTECH INVESTMENTS, INC. (US) 2021-03-25 WO disclosed