SCHEMBL23157263

SCHEMBL23157263

CNc1ncnc(NC(=O)c2ccccc2)c1N

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.51
EGFR P00533 2/20 0.46
AURKB Q96GD4 2/20 0.46
P2RX3 P56373 1/20 0.46
HTT P42858 2/20 0.46
CYP1A2 P05177 1/20 0.46
MAPT P10636 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
HDAC3 O15379 1/20 0.45
MAPK1 P28482 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC2 Q92769 1/20 0.45
CSF1R P07333 1/20 0.44
NT5C2 P49902 2/20 0.44
BCAT2 O15382 1/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
NPSR1 Q6W5P4 1/20 0.43
AURKA O14965 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18521523 0.74 BRD4 (0.52) BRD4EGFRAURKBP2RX3HTT
SCHEMBL5031511 0.72 HDAC3 (0.51) BRD4HDAC3MAPK1HDAC1HDAC2
SCHEMBL27873799 0.72 ADORA3 (0.66) BRD4EGFRAURKBMAPTMAPK1
SCHEMBL23123 0.72 BRD4 (0.64) BRD4EGFRAURKBHTTCSF1R
SCHEMBL23283445 0.72 EGFR (0.76) BRD4EGFRAURKBCSF1RNT5C2
SCHEMBL2343403 0.71 MAPK1 (0.58) BRD4EGFRAURKBMAPK1CSF1R
SCHEMBL8381773 0.71 BRD4 (0.63) BRD4EGFRAURKBHTTCSF1R
SCHEMBL11831465 0.70 MEN1 (0.64) P2RX3HTTCYP1A2MAPTCYP2C9
SCHEMBL14439750 0.70 NPC1 (0.61) HTTHDAC3MAPK1HDAC1HDAC2
SCHEMBL21356268 0.69 BRAF (0.49) BRD4EGFRAURKBHTTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2813512-B1 PEPTIDE-COMPOUND CYCLIZATION METHOD CHUGAI PHARMACEUTICAL CO LTD (JP) 2021-03-31 EP disclosed