SCHEMBL23166350

SCHEMBL23166350

O=C(O)c1ccc2c(c1)Cc1cc(F)ccc1-2

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 5/20 0.67
MAPT P10636 2/20 0.55
NPC1 O15118 1/20 0.55
RAB9A P51151 1/20 0.55
SRD5A1 P18405 4/20 0.53
ALDH1A1 P00352 3/20 0.50
CYP1A2 P05177 2/20 0.50
CYP2C9 P11712 1/20 0.50
HIF1A Q16665 1/20 0.50
HSD17B1 P14061 1/20 0.47
SLC1A3 P43003 1/20 0.47
SLC1A2 P43004 1/20 0.47
SLC1A1 P43005 1/20 0.47
BCL2L1 Q07817 1/20 0.46
BAD Q92934 1/20 0.46
MAPK14 Q16539 1/20 0.45
TDP2 O95551 2/20 0.45
HPGD P15428 1/20 0.44
AKR1C3 P42330 1/20 0.42
DRD2 P14416 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31456551 0.89 SRD5A2 (0.81) SRD5A2MAPTNPC1RAB9ASRD5A1
SCHEMBL27506 0.89 SRD5A2 (0.81) SRD5A2MAPTNPC1RAB9ASRD5A1
SCHEMBL11812488 0.87 NPC1 (0.56) SRD5A2MAPTNPC1RAB9ASRD5A1
Hydrochloric Acid SCHEMBL9789481 0.87 SRD5A2 (0.79) SRD5A2MAPTNPC1RAB9ASRD5A1
SCHEMBL24503134 0.85 SRD5A2 (0.49) SRD5A2MAPTNPC1RAB9ASRD5A1
SCHEMBL1647589 0.83 SRD5A2 (0.79) SRD5A2MAPTNPC1RAB9ASRD5A1
SCHEMBL30976964 0.83 SRD5A2 (0.79) SRD5A2MAPTNPC1RAB9ASRD5A1
SCHEMBL11685606 0.81 MAPK14 (0.60) SRD5A2SRD5A1ALDH1A1MAPK14TTR
SCHEMBL23166496 0.80 MAPT (0.53) SRD5A2MAPTNPC1RAB9AALDH1A1
SCHEMBL577480 0.80 PGR (0.49) MAPTNPC1RAB9ASRD5A1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240269293-A1 PROTEIN-MACROMOLECULE CONJUGATES AND METHODS OF USE THEREOF OD THERAPEUTICS LIMITED (CN) 2024-08-15 US disclosed
EP-4313154-A1 PROTEIN-MACROMOLECULE CONJUGATES AND METHODS OF USE THEREOF OD Therapeutics Limited (HK) 2024-02-07 EP disclosed
CN-117355337-A Protein-macromolecule conjugates and methods of use thereof 奥迪曼药业科技有限公司 2024-01-05 CN disclosed
US-20220401561-A1 PROTEIN-MACROMOLECULE CONJUGATES AND METHODS OF USE THEREOF AJ SCIENCES (YIXING) CO., LTD (CN) 2022-12-22 US disclosed
US-20220401561-A1 PROTEIN-MACROMOLECULE CONJUGATES AND METHODS OF USE THEREOF AJ SCIENCES (YIXING) CO., LTD (CN) 2022-12-22 US disclosed
WO-2022212362-A1 PROTEIN-MACROMOLECULE CONJUGATES AND METHODS OF USE THEREOF BEIJING XUANYI PHARMASCIENCES CO., LTD. (CN) 2022-10-06 WO disclosed
EP-4037715-A1 PROTEIN-MACROMOLECULE CONJUGATES AND METHODS OF USE THEREOF Beijing Xuanyi Pharmasciences Co., Ltd. (CN) 2022-08-10 EP disclosed
CN-114630818-A Protein-macromolecule conjugates and methods of use thereof 北京轩义医药科技有限公司 2022-06-14 CN disclosed
WO-2021067458-A1 PROTEIN-MACROMOLECULE CONJUGATES AND METHODS OF USE THEREOF BEIJING XUANYI PHARMASCIENCES CO., LTD. (CN) 2021-04-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240269293-A1 PROTEIN-MACROMOLECULE CONJUGATES AND METHODS OF USE THEREOF CD44, MACROD1, MSN SRD5A2 4748/4885MAPT 1112/4885NPC1 3707/4885
US-20220401561-A1 PROTEIN-MACROMOLECULE CONJUGATES AND METHODS OF USE THEREOF CD44, SSB, DNPEP SRD5A2 4699/4885MAPT 1431/4885NPC1 3854/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.