SCHEMBL23173151

SCHEMBL23173151

CN1C(=O)CCC(N2Cc3cc(N)ccc3C2=O)C1=O

nearest known ligand 0.61

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 12/20 0.61
CASP1 P29466 1/20 0.40
CASP7 P55210 1/20 0.40
HSD17B10 Q99714 1/20 0.40
IKZF2 Q9UKS7 6/20 0.39
DDB1 Q16531 2/20 0.38
CSNK1A1 P48729 2/20 0.36
CYP19A1 P11511 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22940154 0.90 CRBN (0.68) CRBNDDB1CYP19A1
SCHEMBL24319166 0.86 CRBN (0.60) CRBNIKZF2DDB1CSNK1A1
SCHEMBL26107723 0.85 CRBN (0.58) CRBNIKZF2DDB1CSNK1A1
SCHEMBL31347063 0.85 CRBN (0.58) CRBNIKZF2DDB1CSNK1A1
SCHEMBL26518780 0.84 CRBN (0.58) CRBNCASP1CASP7HSD17B10IKZF2
SCHEMBL27097398 0.83 CRBN (0.59) CRBNIKZF2CSNK1A1
SCHEMBL24745571 0.83 CRBN (0.56) CRBNIKZF2DDB1CSNK1A1
SCHEMBL30121132 0.82 CRBN (0.63) CRBNDDB1
SCHEMBL824532 0.82 CRBN (0.63) CRBNDDB1
SCHEMBL26075169 0.81 CRBN (0.57) CRBNCASP1CASP7IKZF2DDB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230303538-A1 GALECTIN-3 INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2023-09-28 US disclosed
US-20230303538-A1 GALECTIN-3 INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2023-09-28 US disclosed
CN-115768768-A Galectin-3 inhibitors 百时美施贵宝公司 2023-03-07 CN disclosed
WO-2021242982-A1 GALECTIN-3 INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2021-12-02 WO disclosed
WO-2021180103-A1 DEGRADATION OF BRUTON'S TYROSINE KINASE (BTK) BY CONJUGATION OF BTK INHIBITORS WITH E3 LIGASE LIGAND AND METHODS OF USE BEIGENE, LTD. (KY) 2021-09-16 WO disclosed
WO-2021058017-A1 DEGRADATION OF ANDROGEN RECEPTOR (AR) BY CONJUGATION OF AR ANTAGONISTS WITH E3 LIGASE LIGAND AND METHODS OF USE BEIGENE, LTD. (KY) 2021-04-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230303538-A1 GALECTIN-3 INHIBITORS LGALS3, LGALS1, LGALS3BP CRBN 3037/4885CASP1 690/4885CASP7 1158/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.