SCHEMBL2317642

SCHEMBL2317642

CC1(C)C=C(/C=C/C=C/C(=O)O)c2ccccc2OC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MASP2 O00187 1/20 0.37
F2 P00734 1/20 0.37
ESR1 P03372 1/20 0.35
ESR2 Q92731 1/20 0.35
KDM4E B2RXH2 3/20 0.35
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
MAPT P10636 1/20 0.32
PKM P14618 1/20 0.32
MAOB P27338 1/20 0.32
ALOX5 P09917 1/20 0.32
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
NFKB1 P19838 1/20 0.31
CA4 P22748 1/20 0.31
RARA P10276 1/20 0.31
RARB P10826 1/20 0.31
RARG P13631 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1399994 1.00 CYP1A2 (0.39) CYP1A2HSD17B10MASP2F2ESR1
SCHEMBL4948190 0.83 RXRA (0.42) HSD17B10KDM4EALDH1A1MAPTPKM
SCHEMBL3611755 0.83 RXRA (0.42) HSD17B10KDM4EALDH1A1MAPTPKM
SCHEMBL3611761 0.83 RXRA (0.42) HSD17B10KDM4EALDH1A1MAPTPKM
SCHEMBL1400110 0.77 PKM (0.37) PKMMAOB
SCHEMBL2314407 0.71 HTR2B (0.38) ESR1ESR2KDM4EMAPTALOX5
SCHEMBL2314399 0.71 HTR2B (0.38) ESR1ESR2KDM4EMAPTALOX5
SCHEMBL3599366 0.71 RXRA (0.41) HSD17B10KDM4EALDH1A1MAPTPKM
SCHEMBL6859855 0.70 KDM4E (0.42) ESR1ESR2KDM4EALDH1A1HPGD
SCHEMBL3596227 0.69 RAB9A (0.39) KDM4EALDH1A1HPGDMAPTPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1609786-B1 5-alkenone-3,3-dimethyl-benzoxepines derivatives useful for the preparation of antidiabetic pentadienoic acids MERCK SANTE SAS (FR) 2011-08-03 EP disclosed
EP-1609786-A1 New 5-alkenone-3,3-dimethyl-benzoxepines derivatives useful for the preparation of antidiabetic pentadienoic acids Merck Sante (FR) 2005-12-28 EP disclosed