SCHEMBL2318

SCHEMBL2318

CCCCC(=O)N(Cc1ccc(-c2ccccc2C#N)cc1)C1(C(=O)OCc2ccccc2)CCCCC1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.44
LTB4R2 Q9NPC1 14/20 0.43
FFAR1 O14842 1/20 0.42
AKR1B1 P15121 1/20 0.42
OXTR P30559 1/20 0.42
AVPR1A P37288 1/20 0.42
AGTR1 P30556 1/20 0.40
ITGB1 P05556 1/20 0.38
ITGA4 P13612 1/20 0.38
CTSL P07711 1/20 0.38
CTSB P07858 1/20 0.38
CTSS P25774 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3575 0.99 ACHE (0.44) ACHELTB4R2FFAR1AKR1B1OXTR
SCHEMBL3375483 0.86 ACHE (0.47) ACHELTB4R2OXTRAVPR1AAGTR1
SCHEMBL27191042 0.82 LTB4R2 (0.41) ACHELTB4R2AGTR1ITGB1ITGA4
SCHEMBL3077 0.81 LTB4R2 (0.44) LTB4R2AGTR1
SCHEMBL1993 0.80 LTB4R2 (0.45) LTB4R2AGTR1
SCHEMBL21083703 0.80 LTB4R2 (0.41) ACHELTB4R2FFAR1AKR1B1AGTR1
SCHEMBL2366 0.79 LTB4R2 (0.47) ACHELTB4R2FFAR1AKR1B1OXTR
SCHEMBL21083532 0.78 LTB4R2 (0.47) ACHELTB4R2AGTR1
SCHEMBL21083851 0.78 LTB4R2 (0.45) ACHELTB4R2AGTR1
SCHEMBL29726839 0.78 LTB4R2 (0.45) ACHELTB4R2AGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0443983-B1 Acyl compounds CIBA GEIGY AG (CH) 1996-02-28 EP disclosed
US-5399578-A Hypotensive; valsartan; high blood pressure and cardiac insufficiency CIBA-GEIGY CORP (US) 1995-03-21 US disclosed
EP-0443983-A1 Acyl compounds CIBA-GEIGY AG (CH) 1991-08-28 EP disclosed