SCHEMBL2318237

SCHEMBL2318237

O=C(O)C[C@H](CCc1ccccc1)N(C(=O)C1CC1)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.46
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
CTSG P08311 1/20 0.40
CTRB1 P17538 1/20 0.40
OPRM1 P35372 4/20 0.40
CHRM3 P20309 3/20 0.40
CHRM2 P08172 2/20 0.40
MMP12 P39900 2/20 0.40
MMP2 P08253 1/20 0.40
MMP9 P14780 1/20 0.40
MMP13 P45452 1/20 0.40
MMP14 P50281 1/20 0.40
HPGD P15428 1/20 0.39
ADRA1A P35348 3/20 0.38
ADRA1B P35368 3/20 0.38
OPRD1 P41143 3/20 0.38
OPRK1 P41145 3/20 0.38
CHRM1 P11229 2/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2312144 1.00 HTT (0.46) HTTMEN1KMT2ACTSGCTRB1
SCHEMBL4962348 0.73 HTT (0.43) HTTMEN1KMT2AOPRM1CHRM3
SCHEMBL7492223 0.72 HTT (0.39) HTTMEN1KMT2AOPRM1CHRM3
SCHEMBL5871034 0.70 SLC6A2 (0.37) HTTMEN1KMT2ACHRM3CHRM2
SCHEMBL18065715 0.66 MMP12 (0.56) MMP12MMP2MMP9MMP13MMP14
SCHEMBL24726680 0.65 OPRD1 (0.76) OPRM1CHRM3CHRM2ADRA1AADRA1B
SCHEMBL687094 0.65 MMP12 (0.80) MMP12MMP2MMP9MMP13MMP14
SCHEMBL8333817 0.65 MMP12 (0.80) MMP12MMP2MMP9MMP13MMP14
SCHEMBL4745347 0.65 MMP12 (0.80) MMP12MMP2MMP9MMP13MMP14
SCHEMBL27109144 0.65 KEAP1 (0.57) HTTMEN1KMT2AADRA1AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011092284-A1 NOVEL AMINO ACID DERIVATIVES AND THEIR USE AS GPR43 RECEPTOR MODULATORS EUROSCREEN S.A. (BE) 2011-08-04 WO claimed