SCHEMBL23201602

SCHEMBL23201602

COc1ncccc1-c1cccc(C(=O)NC2CN(C)C2)n1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 1/20 0.56
HRH4 Q9H3N8 1/20 0.41
NTRK1 P04629 2/20 0.40
SCN9A Q15858 1/20 0.40
CTSA P10619 3/20 0.40
WDR5 P61964 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
USP30 Q70CQ3 2/20 0.39
PDE4B Q07343 3/20 0.39
PDE4D Q08499 2/20 0.39
MC2R Q01718 2/20 0.39
PDCD1 Q15116 1/20 0.38
CD274 Q9NZQ7 1/20 0.38
KDM1A O60341 1/20 0.38
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30090944 0.84 MC2R (0.54) IRAK4NTRK1USP30MC2R
SCHEMBL30090945 0.84 MC2R (0.54) IRAK4NTRK1USP30MC2R
SCHEMBL31162221 0.84 MC2R (0.54) IRAK4NTRK1USP30MC2R
SCHEMBL31188553 0.77 IRAK4 (0.53) IRAK4ALDH1A1USP30
SCHEMBL31077928 0.75 DGAT2 (0.49) IRAK4NTRK1ALDH1A1MC2R
SCHEMBL30200058 0.74 GRM5 (0.62) NTRK1ALDH1A1
SCHEMBL31077750 0.73 MC2R (0.55) MC2R
SCHEMBL31077853 0.73 USP30 (0.59) USP30MC2R
SCHEMBL12753663 0.73 HSD11B1 (0.64) IRAK4HRH4SCN9AALDH1A1HPGD
SCHEMBL16465114 0.72 IRAK4 (1.00) IRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3802500-A1 MELANOCORTIN SUBTYPE-2 RECEPTOR (MC2R) ANTAGONISTS AND USES THEREOF Crinetics Pharmaceuticals, Inc. (US) 2021-04-14 EP claimed