SCHEMBL23201719

SCHEMBL23201719

COC(=O)c1cc(Br)ccc1N1CCNCC1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 8/20 0.51
KDM4E B2RXH2 2/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
HTR6 P50406 2/20 0.45
HTR7 P34969 1/20 0.45
HTR4 Q13639 1/20 0.45
NR4A2 P43354 1/20 0.45
ALDH1A1 P00352 2/20 0.44
OPRK1 P41145 1/20 0.43
HTR3E A5X5Y0 1/20 0.43
HTR3B O95264 1/20 0.43
HTR3A P46098 1/20 0.43
HTR3D Q70Z44 1/20 0.43
HTR3C Q8WXA8 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL21700700 0.99 BACE1 (0.50) BACE1KDM4EMEN1KMT2AHTR6
SCHEMBL16279248 0.95 BACE1 (0.47) BACE1KDM4EMEN1KMT2AHTR6
SCHEMBL30918477 0.89 KDM4E (0.47) BACE1KDM4EMEN1KMT2AHTR6
SCHEMBL24983954 0.89 KDM4E (0.47) BACE1KDM4EMEN1KMT2AHTR6
SCHEMBL17893724 0.84 ALDH1A1 (0.45) KDM4EMEN1KMT2ANR4A2ALDH1A1
SCHEMBL17916000 0.84 OPRK1 (0.50) KDM4EMEN1KMT2ANR4A2ALDH1A1
SCHEMBL652911 0.83 HTR3E (0.56) KDM4EMEN1KMT2AHTR6HTR7
SCHEMBL19680543 0.83 MAPT (0.56) BACE1KDM4EMEN1KMT2AALDH1A1
SCHEMBL10267394 0.82 ALDH1A1 (0.49) KDM4EMEN1KMT2AHTR6ALDH1A1
SCHEMBL29249371 0.82 KDM4E (0.44) BACE1KDM4EMEN1KMT2AHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3802500-A1 MELANOCORTIN SUBTYPE-2 RECEPTOR (MC2R) ANTAGONISTS AND USES THEREOF Crinetics Pharmaceuticals, Inc. (US) 2021-04-14 EP disclosed