SCHEMBL2320403

SCHEMBL2320403

CCOc1ccc2ccc(Cl)nc2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 5/20 0.53
KMT2A Q03164 2/20 0.51
MAPT P10636 2/20 0.47
NQO1 P15559 1/20 0.45
ALDH1A1 P00352 2/20 0.44
TP53 P04637 1/20 0.44
CYP3A4 P08684 1/20 0.44
TSHR P16473 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CYP1A2 P05177 1/20 0.42
CA4 P22748 1/20 0.42
CA6 P23280 1/20 0.42
CA5A P35218 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
CA14 Q9ULX7 1/20 0.42
CA5B Q9Y2D0 1/20 0.42
CYP11B1 P15538 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2323241 0.88 KMT2A (0.54) NCF1KMT2AMAPTNQO1ALDH1A1
SCHEMBL12957276 0.86 NCF1 (0.54) NCF1KMT2AMAPTALDH1A1CYP3A4
SCHEMBL23452966 0.82 NCF1 (0.74) NCF1MAPTALDH1A1TP53CYP3A4
SCHEMBL20909590 0.80 NCF1 (0.49) NCF1ALDH1A1CYP1A2KDM4E
SCHEMBL13737643 0.80 MAPT (0.53) NCF1KMT2AMAPTNQO1ALDH1A1
SCHEMBL622376 0.79 ALDH1A1 (0.56) NCF1KMT2ANQO1ALDH1A1HSD17B10
SCHEMBL20909360 0.79 NCF1 (0.51) NCF1ALDH1A1CYP3A4KDM4E
SCHEMBL28158822 0.79 CA12 (0.48) NCF1KMT2AMAPTALDH1A1CA12
SCHEMBL29205379 0.79 NCF1 (0.48) NCF1ALDH1A1KDM4E
SCHEMBL17430103 0.78 ALDH1A1 (0.41) NCF1KMT2AMAPTALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 36 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2531032-B1 MATERIALS AND METHOD FOR INHIBITING REPLICATION PROTEIN A AND USES THEREOF UNIV INDIANA RES & TECH CORP (US) 2019-04-10 EP claimed
CN-105037266-A Antibacterial chloroxoquinoline derivative WANG ZIHOU 2015-11-11 CN claimed
CN-105017145-A Chloroxoquinoline derivative with anti-tumor activity WANG ZIHOU 2015-11-04 CN claimed
US-20140370121-A1 MATERIALS AND METHOD FOR INHIBITING REPLICATION PROTEIN A AND USES THEREOF INDIANA UNIVERSITY RESEARCH & TECHNOLOGY CORPORATION 2014-12-18 US claimed
US-8859532-B2 Materials and method for inhibiting replication protein A and uses thereof INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORP. (US) 2014-10-14 US claimed
CN-103864681-A Chloroxoquinoline derivatives for antibacterial use WANG ZIHOU 2014-06-18 CN claimed
CN-103864680-A Chloroxoquinoline derivative with antineoplastic activity WANG ZIHOU 2014-06-18 CN claimed
US-20130028989-A1 MATERIALS AND METHOD FOR INHIBITING REPLICATION PROTEIN A AND USES THEREOF INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORATION (US) 2013-01-31 US claimed
EP-2531032-A1 MATERIALS AND METHOD FOR INHIBITING REPLICATION PROTEIN A AND USES THEREOF Indiana University Research and Technology Corporation (US) 2012-12-12 EP claimed
WO-2011097545-A9 MATERIALS AND METHOD FOR INHIBITING REPLICATION PROTEIN A AND USES THEREOF INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORTION (US) 2011-11-17 WO claimed
WO-2011097545-A1 MATERIALS AND METHOD FOR INHIBITING REPLICATION PROTEIN A AND USES THEREOF INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORTION (US) 2011-08-11 WO claimed
US-20220153747-A1 Selective Inhibitors Of Protein Arginine Methytransterase 5 (PRMT5) PRELUDE THERAPEUTICS, INCORPORATED 2022-05-19 US disclosed
US-11208416-B2 Selective inhibitors of protein arginine methytransterase 5 (PRMT5) PRELUDE THERAPEUTICS INCORPORATED (US) 2021-12-28 US disclosed
US-20200361946-A1 Selective Inhibitors Of Protein Arginine Methytransterase 5 (PRMT5) PRELUDE THERAPEUTICS INC (US) 2020-11-19 US disclosed
EP-2531032-B1 MATERIALS AND METHOD FOR INHIBITING REPLICATION PROTEIN A AND USES THEREOF UNIV INDIANA RES & TECH CORP (US) 2019-04-10 EP disclosed
CN-103588755-A Preparation method for neratinib CHIA TAI TIANQING PHARMACEUTICAL GROUP CO LTD 2014-02-19 CN disclosed
US-20130028989-A1 MATERIALS AND METHOD FOR INHIBITING REPLICATION PROTEIN A AND USES THEREOF INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORATION (US) 2013-01-31 US disclosed
EP-2531032-A1 MATERIALS AND METHOD FOR INHIBITING REPLICATION PROTEIN A AND USES THEREOF Indiana University Research and Technology Corporation (US) 2012-12-12 EP disclosed
WO-2011097545-A9 MATERIALS AND METHOD FOR INHIBITING REPLICATION PROTEIN A AND USES THEREOF INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORTION (US) 2011-11-17 WO disclosed
WO-2011097545-A1 MATERIALS AND METHOD FOR INHIBITING REPLICATION PROTEIN A AND USES THEREOF INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORTION (US) 2011-08-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140370121-A1 MATERIALS AND METHOD FOR INHIBITING REPLICATION PROTEIN A AND USES THEREOF RPA1, RPA3, PCNA NCF1 1321/4885KMT2A 1671/4885MAPT 4175/4885
US-20130028989-A1 MATERIALS AND METHOD FOR INHIBITING REPLICATION PROTEIN A AND USES THEREOF RPA1, RPA3, PCNA NCF1 1321/4885KMT2A 1671/4885MAPT 4175/4885
US-11208416-B2 Selective inhibitors of protein arginine methytransterase 5 (PRMT5) PRMT5, PRMT1, PRMT6 NCF1 1771/4885KMT2A 409/4885MAPT 1824/4885
US-20220153747-A1 Selective Inhibitors Of Protein Arginine Methytransterase 5 (PRMT5) PRMT5, PRMT1, PRMT6 NCF1 1771/4885KMT2A 409/4885MAPT 1824/4885
US-20200361946-A1 Selective Inhibitors Of Protein Arginine Methytransterase 5 (PRMT5) PRMT5, PRMT1, PRMT6 NCF1 1771/4885KMT2A 409/4885MAPT 1824/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.