SCHEMBL23212930

SCHEMBL23212930

Cc1ccc(S(=O)(=O)OCCC(CCOS(=O)(=O)c2ccc(C)cc2)c2ccccc2Br)cc1.OCCC(CCO)c1ccccc1Br

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.36
KMT2A Q03164 3/20 0.36
POLB P06746 2/20 0.36
CYP24A1 Q07973 1/20 0.35
DHODH Q02127 1/20 0.34
VDR P11473 1/20 0.34
CYP3A4 P08684 3/20 0.34
LMNA P02545 2/20 0.34
MAPK1 P28482 2/20 0.34
CYP2D6 P10635 2/20 0.34
THPO P40225 1/20 0.34
STAT3 P40763 1/20 0.34
MEN1 O00255 2/20 0.34
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA9 Q16790 1/20 0.33
CYP2C19 P33261 3/20 0.33
ALOX15 P16050 1/20 0.33
KEAP1 Q14145 1/20 0.32
NFE2L2 Q16236 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23210214 0.94 VDR (0.38) ALDH1A1KMT2APOLBCYP24A1DHODH
SCHEMBL23212923 0.84 PSEN1 (0.38) ALDH1A1KMT2ALMNACYP2D6STAT3
SCHEMBL23212936 0.81 RORC (0.35) ALDH1A1KMT2AVDRLMNAMAPK1
SCHEMBL23213256 0.79 CFTR (0.37) ALDH1A1CYP3A4LMNACYP2D6CA12
SCHEMBL29843909 0.77 CA12 (0.36) ALDH1A1KMT2AVDRCYP3A4MAPK1
SCHEMBL23210189 0.77 CA12 (0.36) ALDH1A1KMT2AVDRCYP3A4MAPK1
SCHEMBL2537530 0.76 DHODH (0.40) ALDH1A1KMT2APOLBDHODHVDR
SCHEMBL7840144 0.75 ALDH1A1 (0.43) ALDH1A1CYP24A1VDRCYP3A4LMNA
SCHEMBL3940918 0.75 STAT3 (0.40) ALDH1A1KMT2APOLBCYP2D6STAT3
SCHEMBL3940922 0.75 STAT3 (0.40) ALDH1A1KMT2APOLBCYP2D6STAT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021070091-A1 5-OXA-2-AZASPIRO[3.4]OCTANE DERIVATIVES AS M4 AGONISTS NOVARTIS AG (CH) 2021-04-15 WO disclosed
WO-2021070090-A1 2-AZASPIRO[3.4]OCTANE DERIVATIVES AS M4 AGONISTS NOVARTIS AG (CH) 2021-04-15 WO disclosed