SCHEMBL23213849

SCHEMBL23213849

Cc1c(Cl)cc(N)cc1CN1CC2(COC2)C1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 1/20 0.38
CD274 Q9NZQ7 1/20 0.38
GSPT1 P15170 1/20 0.37
CRBN Q96SW2 1/20 0.37
CYP1A2 P05177 1/20 0.32
CHRM4 P08173 1/20 0.32
ADCY10 Q96PN6 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
TLR8 Q9NR97 1/20 0.31
TLR7 Q9NYK1 1/20 0.31
SCN1A P35498 1/20 0.31
SCN5A Q14524 1/20 0.31
SCN8A Q9UQD0 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
CYP2A13 Q16696 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29796045 1.00 PDCD1 (0.38) PDCD1CD274GSPT1CRBNCYP1A2
SCHEMBL29796043 1.00 PDCD1 (0.38) PDCD1CD274GSPT1CRBNCYP1A2
SCHEMBL27290054 0.86 CD274 (0.39) PDCD1CD274GSPT1CRBNCYP1A2
SCHEMBL23240233 0.83 CD274 (0.36) PDCD1CD274ADCY10TLR8TLR7
SCHEMBL29739690 0.78 CYP2A13 (0.51) MAPTSMN1; SMN2TDP1CYP2A13
SCHEMBL23213276 0.78 CYP2A13 (0.51) MAPTSMN1; SMN2TDP1CYP2A13
SCHEMBL23213311 0.78 LMNA (0.40) PDCD1CD274GSPT1CRBNALDH1A1
SCHEMBL29795970 0.78 LMNA (0.40) PDCD1CD274GSPT1CRBNALDH1A1
SCHEMBL23213302 0.77 GSPT1 (0.49) PDCD1CD274GSPT1CRBNSCN1A
SCHEMBL23213589 0.74 LMNA (0.50) CYP1A2ALDH1A1MAPTSMN1; SMN2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240216355-A1 PHARMACEUTICAL COMPOSITIONS FOR USE IN THE PREVENTION AND TREATMENT OF A DISEASE OR DISORDER CAUSED BY OR ASSOCIATED WITH ONE OR MORE PREMATURE TERMINATION CODONS MONTE ROSA THERAPEUTICS AG (CH) 2024-07-04 US disclosed
EP-4313047-A1 PHARMACEUTICAL COMPOSITIONS FOR USE IN THE PREVENTION AND TREATMENT OF A DISEASE OR DISORDER CAUSED BY OR ASSOCIATED WITH ONE OR MORE PREMATURE TERMINATION CODONS Monte Rosa Therapeutics, Inc. (US) 2024-02-07 EP disclosed
US-20220242846-A1 ISOINDOLINONE COMPOUNDS MONTE ROSA THERAPEUTICS AG (CH) 2022-08-04 US disclosed
WO-2021069705-A1 ISOINDOLINONE COMPOUNDS MONTE ROSA THERAPEUTICS (CH) 2021-04-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240216355-A1 PHARMACEUTICAL COMPOSITIONS FOR USE IN THE PREVENTION AND TREATMENT OF A DISEASE OR DISORDER CAUSED BY OR ASSOCIATED WITH ONE OR MORE PREMATURE TERMINATION CODONS UPF1, NSUN2, RTF2 PDCD1 4754/4885CD274 4873/4885GSPT1 1795/4885
US-20220242846-A1 ISOINDOLINONE COMPOUNDS AOC2, AOC3, INF2 PDCD1 3567/4885CD274 3905/4885GSPT1 4622/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.