SCHEMBL23217370

SCHEMBL23217370

NC(=O)C(O)CCCNC(=O)Nc1ccc(S(=O)(=O)N2CCN(c3cc(Cl)cc(C(F)(F)F)c3)CC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.47
CA2 P00918 2/20 0.47
CA7 P43166 1/20 0.47
NAMPT P43490 6/20 0.46
EPHX2 P34913 3/20 0.45
PTGDR Q13258 1/20 0.43
MAPT P10636 2/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
ATM Q13315 1/20 0.41
F13A1 P00488 1/20 0.41
TGM2 P21980 1/20 0.41
TGM1 P22735 1/20 0.41
TRPV4 Q9HBA0 3/20 0.40
TP53 P04637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23217124 0.85 PTPN11 (0.49) CA1CA2CA7NAMPTEPHX2
SCHEMBL23217375 0.84 NAMPT (0.47) CA1CA2CA7NAMPTEPHX2
SCHEMBL23217373 0.84 EPHX2 (0.47) CA1CA2CA7NAMPTEPHX2
SCHEMBL23217109 0.83 NAMPT (0.47) CA1CA2CA7NAMPTEPHX2
SCHEMBL23217303 0.79 NAMPT (0.44) CA1CA2CA7NAMPTEPHX2
SCHEMBL25381894 0.78 MAPT (0.66) EPHX2MAPTKDM4EALDH1A1ATM
SCHEMBL30563199 0.78 MAPT (0.66) EPHX2MAPTKDM4EALDH1A1ATM
SCHEMBL25380430 0.76 TRPV4 (0.55) PTGDRMAPTALDH1A1TRPV4
SCHEMBL31252083 0.75 TRPV4 (0.58) MAPTKDM4EALDH1A1F13A1TGM2
SCHEMBL23217265 0.75 PTPN11 (0.56) CA1CA2CA7NAMPTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021072369-A1 LPXH TARGETING COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF MAKING AND USING THE SAME DUKE UNIVERSITY (US) 2021-04-15 WO disclosed