SCHEMBL23218007

SCHEMBL23218007

Cc1cccc(-c2n[nH]cc2-c2ccc(F)c(-c3cnn(CCN4C(=O)c5ccccc5C4=O)c3)c2)n1

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 12/20 0.54
FEN1 P39748 3/20 0.36
ALDH1A1 P00352 1/20 0.34
MAP3K5 Q99683 2/20 0.33
MAPK14 Q16539 2/20 0.33
CHRM1 P11229 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23218015 0.88 TGFBR1 (0.59) TGFBR1FEN1MAPK14
SCHEMBL29361356 0.87 TGFBR1 (0.70) TGFBR1FEN1MAPK14
SCHEMBL5198271 0.87 TGFBR1 (0.70) TGFBR1FEN1MAPK14
SCHEMBL5199498 0.86 TGFBR1 (0.56) TGFBR1MAPK14
SCHEMBL5198295 0.85 TGFBR1 (0.56) TGFBR1FEN1MAP3K5
SCHEMBL5200014 0.84 TGFBR1 (0.53) TGFBR1
SCHEMBL24311917 0.84 TGFBR1 (0.56) TGFBR1MAPK14
SCHEMBL5198228 0.83 TGFBR1 (0.52) TGFBR1FEN1MAPK14
SCHEMBL24311918 0.82 TGFBR1 (0.53) TGFBR1MAPK14
SCHEMBL24311947 0.82 TGFBR1 (0.53) TGFBR1MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022076905-A1 ALK5 INHIBITORS, CONJUGATES, AND USES THEREOF SILVERBACK THERAPEUTICS, INC. (US) 2022-04-14 WO disclosed
WO-2021072330-A1 GALNAC-TGFBR1 INHIBITOR CONJUGATES FOR THE TREATMENT OF LIVER DISEASES SILVERBACK THERAPEUTICS, INC. (US) 2021-04-15 WO disclosed