SCHEMBL23218441

SCHEMBL23218441

CCOC(=O)Cc1ccccc1OCc1csc2ccc(Cl)cc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.49
NFE2L2 Q16236 1/20 0.49
PTGDR2 Q9Y5Y4 1/20 0.45
MAPT P10636 2/20 0.43
PPARD Q03181 2/20 0.42
PPARA Q07869 2/20 0.42
PPARG P37231 1/20 0.42
CYP2A6 P11509 3/20 0.41
TBXAS1 P24557 1/20 0.41
PKM P14618 1/20 0.40
EGFR P00533 1/20 0.40
ERBB2 P04626 1/20 0.40
EPHA2 P29317 1/20 0.40
KDR P35968 1/20 0.40
EPHB4 P54760 1/20 0.40
CFD P00746 1/20 0.40
SLC22A12 Q96S37 1/20 0.39
FFAR4 Q5NUL3 1/20 0.39
PTGER1 P34995 1/20 0.39
NPC1 O15118 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29853164 1.00 KEAP1 (0.49) KEAP1NFE2L2PTGDR2MAPTPPARD
SCHEMBL28566073 0.85 KEAP1 (0.66) KEAP1NFE2L2MAPTCYP2A6SLC22A12
SCHEMBL29853072 0.81 CFD (0.56) PPARDPPARAPPARGTBXAS1CFD
SCHEMBL23218062 0.81 CFD (0.56) PPARDPPARAPPARGTBXAS1CFD
SCHEMBL2350834 0.74 SLC22A12 (0.44) KEAP1NFE2L2MAPTCYP2A6SLC22A12
SCHEMBL29852542 0.74 PTGDR2 (0.39) PTGDR2MAPTTBXAS1PKMCFD
SCHEMBL23218713 0.74 PTGDR2 (0.39) PTGDR2MAPTTBXAS1PKMCFD
SCHEMBL31164737 0.74 MTNR1A (0.54) KEAP1NFE2L2MAPTPKM
SCHEMBL10982992 0.74 MTNR1A (0.54) KEAP1NFE2L2MAPTPKM
SCHEMBL8249919 0.73 MAPT (0.43) KEAP1NFE2L2PTGDR2MAPTCYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12558341-B2 Oral complement factor D inhibitors BIOCRYST PHARMACEUTICALS, INC. (US) 2026-02-24 US disclosed
US-20250186391-A1 ORAL COMPLEMENT FACTOR D INHIBITORS WILMINGTON TRUST, NATIONAL ASSOCIATION 2025-06-12 US disclosed
EP-4041238-A1 ORAL COMPLEMENT FACTOR D INHIBITORS Biocryst Pharmaceuticals, Inc. (US) 2022-08-17 EP disclosed
CN-114502168-A Oral complement factor D inhibitors 拜奥克里斯特制药公司 2022-05-13 CN disclosed
WO-2021072198-A1 ORAL COMPLEMENT FACTOR D INHIBITORS BIOCRYST PHARMACEUTICALS, INC. (US) 2021-04-15 WO disclosed
WO-2021072198-A1 ORAL COMPLEMENT FACTOR D INHIBITORS BIOCRYST PHARMACEUTICALS, INC. (US) 2021-04-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12558341-B2 Oral complement factor D inhibitors CFD, CFH, CFB KEAP1 1521/4885NFE2L2 933/4885PTGDR2 484/4885
US-20250186391-A1 ORAL COMPLEMENT FACTOR D INHIBITORS CFD, CFH, CFB KEAP1 1155/4885NFE2L2 925/4885PTGDR2 976/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.