SCHEMBL23219181

SCHEMBL23219181

CC(C)n1nc(COc2cccc(C(=O)O)c2)c2cc(-c3cccc(CN)c3)ccc21

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 8/20 0.50
PLAU P00749 1/20 0.46
MRGPRX4 Q96LA9 5/20 0.45
CFD P00746 1/20 0.43
SSTR5 P35346 1/20 0.43
LOXL2 Q9Y4K0 1/20 0.42
NR1H4 Q96RI1 1/20 0.39
NR4A1 P22736 1/20 0.39
NR4A3 Q92570 1/20 0.39
F2 P00734 1/20 0.39
SRD5A2 P31213 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29591762 1.00 NR4A2 (0.50) NR4A2PLAUMRGPRX4CFDSSTR5
SCHEMBL29852680 0.91 LOXL2 (0.46) NR4A2PLAUMRGPRX4CFDSSTR5
SCHEMBL23218806 0.91 LOXL2 (0.46) NR4A2PLAUMRGPRX4CFDSSTR5
SCHEMBL23218710 0.89 CFD (0.50) NR4A2PLAUCFDSSTR5NR1H4
SCHEMBL23218903 0.86 CFD (0.42) PLAUCFDSSTR5
SCHEMBL23219231 0.84 PLG (0.46) PLAUCFDF2
SCHEMBL28736134 0.82 MRGPRX4 (0.48) NR4A2MRGPRX4SSTR5NR4A1NR4A3
SCHEMBL29592507 0.81 CFD (0.46) PLAUCFD
SCHEMBL23218914 0.81 CFD (0.46) PLAUCFD
SCHEMBL23219211 0.81 CFD (0.62) PLAUCFDF2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4041238-A1 ORAL COMPLEMENT FACTOR D INHIBITORS Biocryst Pharmaceuticals, Inc. (US) 2022-08-17 EP disclosed
CN-114502168-A Oral complement factor D inhibitors 拜奥克里斯特制药公司 2022-05-13 CN disclosed
WO-2021072198-A1 ORAL COMPLEMENT FACTOR D INHIBITORS BIOCRYST PHARMACEUTICALS, INC. (US) 2021-04-15 WO disclosed
WO-2021072198-A1 ORAL COMPLEMENT FACTOR D INHIBITORS BIOCRYST PHARMACEUTICALS, INC. (US) 2021-04-15 WO disclosed