SCHEMBL23255281

SCHEMBL23255281

N#Cc1cc(C#N)cc(-c2ccc3c(c2)c2ccccc2n3-c2ccc(C(F)(F)F)cc2-c2ccncc2-n2c3ccccc3c3cc(-c4cc(C#N)cc(C#N)c4)ccc32)c1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 3/20 0.35
CYP1A2 P05177 2/20 0.34
METAP2 P50579 2/20 0.34
CYP3A4 P08684 2/20 0.33
CYP3A5 P20815 2/20 0.33
KIF11 P52732 2/20 0.32
RXRA P19793 1/20 0.32
RXRG P48443 1/20 0.32
CYP11B2 P19099 1/20 0.31
GRIN1 Q05586 2/20 0.31
GRIN2B Q13224 2/20 0.31
PTPN5 P54829 1/20 0.31
PDE10A Q9Y233 1/20 0.31
EPHX2 P34913 1/20 0.30
NPY5R Q15761 1/20 0.30
PTGDR2 Q9Y5Y4 1/20 0.30
MAT2A P31153 1/20 0.30
CYP11B1 P15538 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23255283 0.95 CYP1A2 (0.35) GPBAR1CYP1A2METAP2CYP3A4CYP3A5
SCHEMBL23255598 0.94 GPBAR1 (0.35) GPBAR1CYP1A2METAP2CYP3A4CYP3A5
SCHEMBL23255282 0.94 KIF11 (0.39) GPBAR1CYP1A2METAP2CYP3A4CYP3A5
SCHEMBL23255315 0.94 CYP1A2 (0.35) GPBAR1CYP1A2METAP2CYP3A4CYP3A5
SCHEMBL23255596 0.90 GPBAR1 (0.33) GPBAR1CYP1A2METAP2CYP3A4CYP3A5
SCHEMBL23255602 0.89 RXRA (0.34) GPBAR1CYP1A2METAP2CYP3A4CYP3A5
SCHEMBL23255587 0.89 CYP3A4 (0.38) GPBAR1CYP1A2METAP2CYP3A4CYP3A5
SCHEMBL21758733 0.89 GPBAR1 (0.35) GPBAR1CYP1A2METAP2CYP3A4CYP3A5
SCHEMBL23255316 0.88 CYP1A2 (0.35) GPBAR1CYP1A2METAP2CYP3A4CYP3A5
SCHEMBL23255279 0.88 KIF11 (0.43) CYP1A2METAP2CYP3A4CYP3A5KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3581570-B1 CARBAZOLE-PYRIDINE-TRIFLUOROMETHYLPHENYL DERIVATIVES AND RELATED COMPOUNDS FOR USE AS TADF LUMINESCENT EMITTERS IN OLEDS CYNORA GMBH (DE) 2021-04-21 EP disclosed