SCHEMBL2327644

SCHEMBL2327644

CC(=O)c1ccc(Cn2nc(C(N)=O)c(-c3nc(C(=O)O)c(-c4cccc(OC(F)(F)F)c4)o3)n2)o1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.39
IRAK4 Q9NWZ3 1/20 0.38
IKBKB O14920 1/20 0.38
HDAC1 Q13547 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
FPR2 P25090 1/20 0.37
FFAR1 O14842 1/20 0.36
FFAR4 Q5NUL3 1/20 0.36
SLC16A3 O15427 1/20 0.36
SLC16A1 P53985 1/20 0.36
MCTS1 Q9ULC4 1/20 0.36
DHODH Q02127 2/20 0.36
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35
DYRK1A Q13627 1/20 0.34
CSNK1D P48730 1/20 0.34
CSNK1E P49674 1/20 0.34
GCGR P47871 1/20 0.34
ATR Q13535 1/20 0.34
LDHA P00338 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2327049 0.91 IKBKB (0.48) ADORA2AIKBKBMAPT
SCHEMBL2327731 0.88 RXRA (0.41) IKBKBHDAC1HDAC6FPR2
SCHEMBL2332690 0.88 NR4A1 (0.37) ADORA2AIKBKBHCRTR1HCRTR2
SCHEMBL2328930 0.87 HCRTR1 (0.44) ADORA2AIKBKBFPR2HCRTR1HCRTR2
SCHEMBL2323238 0.87 IKBKB (0.40) ADORA2AIKBKBHCRTR1HCRTR2
SCHEMBL2331266 0.86 IKBKB (0.45) ADORA2AIKBKBHCRTR1HCRTR2
SCHEMBL2328104 0.86 HCRTR1 (0.36) ADORA2AIKBKBHCRTR1HCRTR2
SCHEMBL2328920 0.86 IKBKB (0.35) ADORA2AIKBKBSLC16A3SLC16A1MCTS1
SCHEMBL2330683 0.85 ADORA2A (0.38) ADORA2AIRAK4IKBKBFPR2FFAR1
SCHEMBL2327570 0.85 LRRK2 (0.36) ADORA2AIKBKBSLC16A3SLC16A1MCTS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2225231-B1 AMINOTRIAZOLE DERIVATIVES AS ALX AGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2011-08-17 EP claimed
EP-2225231-B1 AMINOTRIAZOLE DERIVATIVES AS ALX AGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2011-08-17 EP disclosed