SCHEMBL23280356

SCHEMBL23280356

CN1CCC(Oc2cc(C(=O)O)ccn2)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM2B Q8NHM5 3/20 0.54
GSK3B P49841 3/20 0.52
DYRK1A Q13627 3/20 0.52
WNT1 P04628 2/20 0.52
PRMT5 O14744 3/20 0.45
OPRK1 P41145 1/20 0.45
KCNH2 Q12809 1/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
JMJD6 Q6NYC1 1/20 0.45
KDM4E B2RXH2 2/20 0.43
KDM6B O15054 2/20 0.43
KDM5C P41229 2/20 0.43
KDM4C Q9H3R0 2/20 0.43
KDM2A Q9Y2K7 2/20 0.43
KDM3A Q9Y4C1 2/20 0.43
KDM1A O60341 1/20 0.43
LNPEP Q9UIQ6 1/20 0.43
KDM4A O75164 1/20 0.42
SCN1A P35498 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23062923 0.87 KDM4C (0.49) KDM2BOPRK1KCNH2KDM4EKDM6B
SCHEMBL17572955 0.87 PRMT5 (0.55) PRMT5OPRK1KCNH2KDM4EKDM6B
SCHEMBL19473383 0.86 KDM1A (0.45) KDM2BGSK3BDYRK1AWNT1PRMT5
SCHEMBL17559414 0.85 PRMT5 (0.46) GSK3BDYRK1AWNT1PRMT5OPRK1
SCHEMBL30281322 0.84 LOX (0.49) OPRK1KCNH2KMT2AKDM4EKDM6B
SCHEMBL17572116 0.82 GPR119 (0.53)
SCHEMBL19460867 0.82 GPR119 (0.51) PRMT5
SCHEMBL30578274 0.82 KDM2B (0.58) KDM2BJMJD6KDM4EKDM6BKDM5C
SCHEMBL19473358 0.81 OPRK1 (0.41) KDM2BGSK3BDYRK1AWNT1PRMT5
SCHEMBL17572814 0.81 WNT1 (0.48) KDM2BGSK3BDYRK1AWNT1PRMT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3189041-B1 TETRAHYDROISOQUINOLINE DERIVED PRMT5-INHIBITORS CTXT PTY LTD (AU) 2021-04-28 EP disclosed