SCHEMBL23287166

SCHEMBL23287166

N#Cc1ccc(COc2cc(Br)ccc2F)c(F)c1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 3/20 0.44
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
CCR5 P51681 3/20 0.40
SLC6A4 P31645 1/20 0.40
PRMT5 O14744 1/20 0.39
EGFR P00533 1/20 0.39
PTGER1 P34995 2/20 0.38
USP28 Q96RU2 1/20 0.38
MTNR1B P49286 1/20 0.36
NAAA Q02083 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31425070 1.00 MAPK14 (0.44) MAPK14NPC1RAB9ACCR5SLC6A4
SCHEMBL23273445 0.83 HPD (0.43) MAPK14NPC1RAB9ACCR5PTGER1
SCHEMBL29737930 0.83 HPD (0.43) MAPK14NPC1RAB9ACCR5PTGER1
SCHEMBL29825377 0.81 MAPK14 (0.47) MAPK14PRMT5EGFRPTGER1
SCHEMBL23286936 0.81 MAPK14 (0.47) MAPK14PRMT5EGFRPTGER1
SCHEMBL24320312 0.80 PTGER1 (0.48) MAPK14CCR5PTGER1
SCHEMBL29664227 0.80 MAOB (0.50) MAPK14NPC1RAB9A
SCHEMBL23362070 0.80 MAOB (0.50) MAPK14NPC1RAB9A
SCHEMBL23286738 0.78 NPC1 (0.40) MAPK14NPC1RAB9APRMT5EGFR
SCHEMBL23286794 0.78 MAOB (0.40) MAPK14NPC1RAB9APRMT5EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11702404-B2 GLP-1R modulating compounds GILEAD SCIENCES, INC. (US) 2023-07-18 US disclosed
US-11702404-B2 GLP-1R modulating compounds GILEAD SCIENCES, INC. (US) 2023-07-18 US disclosed
US-20210171499-A1 GLP-1R MODULATING COMPOUNDS GILEAD SCIENCES, INC. 2021-06-10 US disclosed
WO-2021081207-A1 GLP-1R MODULATING COMPOUNDS GILEAD SCIENCES, INC. (US) 2021-04-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11702404-B2 GLP-1R modulating compounds GLP1R, GIPR, GPR119 MAPK14 2254/4885NPC1 1188/4885RAB9A 478/4885
US-20210171499-A1 GLP-1R MODULATING COMPOUNDS GLP1R, GIPR, GPR119 MAPK14 2254/4885NPC1 1188/4885RAB9A 478/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.