SCHEMBL23302001

SCHEMBL23302001

O=C(O)CCCCCCCC(=O)N1CC[C@H](Nc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)C1

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 13/20 0.55
CRBN Q96SW2 13/20 0.55
HDAC1 Q13547 4/20 0.49
HDAC2 Q92769 4/20 0.49
HDAC3 O15379 3/20 0.49
NCOR2 Q9Y618 3/20 0.49
TNF P01375 1/20 0.48
IL1B P01584 1/20 0.48
TBXA2R P21731 1/20 0.48
IKZF1 Q13422 1/20 0.48
IKZF3 Q9UKT9 1/20 0.48
PARP1 P09874 2/20 0.48
STAT3 P40763 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29942621 1.00 DDB1 (0.55) DDB1CRBNHDAC1HDAC2HDAC3
SCHEMBL25036293 0.88 DDB1 (0.58) DDB1CRBNHDAC1HDAC2HDAC3
SCHEMBL23768486 0.82 CRBN (0.55) DDB1CRBNTNFIL1BTBXA2R
SCHEMBL22834201 0.82 CRBN (0.68) DDB1CRBNHDAC1HDAC2HDAC3
SCHEMBL21333201 0.82 CRBN (0.68) DDB1CRBNHDAC1HDAC2HDAC3
SCHEMBL22326316 0.82 CRBN (0.68) DDB1CRBNHDAC1HDAC2HDAC3
SCHEMBL23772794 0.82 DDB1 (0.69) DDB1CRBNHDAC1HDAC2HDAC3
SCHEMBL20142514 0.82 CRBN (0.68) DDB1CRBNHDAC1HDAC2HDAC3
SCHEMBL22325167 0.82 CRBN (0.68) DDB1CRBNHDAC1HDAC2HDAC3
SCHEMBL20242552 0.82 CRBN (0.68) DDB1CRBNHDAC1HDAC2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114728936-A Bifunctional compounds for the treatment of cancer 豪夫迈·罗氏有限公司 2022-07-08 CN disclosed
WO-2021083949-A1 BIFUNCTIONAL COMPOUNDS FOR THE TREATMENT OF CANCER F. HOFFMANN-LA ROCHE AG (CH) 2021-05-06 WO disclosed