SCHEMBL2332912

SCHEMBL2332912

CC(C(=O)O)C(C)(C)CBr

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.36
TP53 P04637 1/20 0.35
ALDH1A1 P00352 2/20 0.35
TSHR P16473 2/20 0.35
GABRR1 P24046 2/20 0.31
RNPEP Q9H4A4 1/20 0.31
MAPT P10636 1/20 0.31
PTGS1 P23219 1/20 0.31
SLC7A5 Q01650 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15040910 0.77 CYP1A2 (0.37) CYP1A2TP53ALDH1A1GABRR1RNPEP
SCHEMBL1572639 0.77 CYP1A2 (0.37) CYP1A2TP53ALDH1A1GABRR1RNPEP
SCHEMBL7960610 0.75 HMGCR (0.46) CYP1A2TP53TSHR
SCHEMBL10954165 0.75 CYP1A2 (0.36) CYP1A2TP53ALDH1A1TSHRGABRR1
Ammonia Solution, Strong SCHEMBL8858444 0.73 HMGCR (0.44) CYP1A2TP53TSHR
SCHEMBL5517726 0.73 FFAR1 (0.43) CYP1A2TP53
Ammonia Solution, Strong SCHEMBL8858449 0.73 HMGCR (0.44) CYP1A2TP53TSHR
SCHEMBL16331317 0.73 ADRA1A (0.37) CYP1A2TP53ALDH1A1TSHR
SCHEMBL21052347 0.71 CYP1A2 (0.48) CYP1A2ALDH1A1
SCHEMBL19262058 0.71 CYP1A2 (0.33) CYP1A2TP53SLC7A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0853618-B1 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N- (AMINOIMINOMETHYL)PHENYLALKYL -AZAHETEROCYCLYLAMIDE COMPOUNDS AVENTIS PHARMA INC (US) 2011-08-17 EP disclosed
EP-0853618-A4 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N- (AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLYLAMIDE COMPOUNDS RHONE POULENC RORER PHARMA (US) 2000-03-15 EP disclosed
US-5958918-A Substituted (sulfinic acid, sulfonic acid, sulfonylamino or sulfinylamino) N- (aminominomethyl)phenylalkyl!-azaheterocyclylamide compounds RHONE-POULENC RORER PHARMACEUTICALS INC. 1999-09-28 US disclosed
EP-0853618-A1 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N- (AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLYLAMIDE COMPOUNDS RHONE-POULENC RORER PHARMACEUTICALS, INC. (US) 1998-07-22 EP disclosed
WO-1996040679-A1 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N-[(AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLYLAMIDE COMPOUNDS RHÔNE-POULENC RORER PHARMACEUTICALS INC. (US) 1996-12-19 WO disclosed