SCHEMBL23329196

SCHEMBL23329196

CC(C)c1ccc2nc(CC(C)c3ccc4c(c3)CCNC4=O)[nH]c2c1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PARP11 Q9NR21 8/20 0.41
PARP10 Q53GL7 7/20 0.41
KDM4E B2RXH2 1/20 0.37
MAPT P10636 1/20 0.37
RPS6KA2 Q15349 1/20 0.36
SCN10A Q9Y5Y9 2/20 0.36
PRF1 P14222 1/20 0.35
GRM5 P41594 5/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL279822 0.78 PARP10 (0.63) PARP11PARP10GRM5
SCHEMBL20132703 0.72 KMT2A (0.46) KDM4EMAPTSCN10A
SCHEMBL25795405 0.71 PARP11 (0.51) PARP11PARP10GRM5
SCHEMBL26353996 0.70 KDM4E (0.42) KDM4EMAPTSCN10A
SCHEMBL5989076 0.68 DDAH1 (0.54) KDM4EMAPTSCN10A
SCHEMBL2611066 0.68 PARP10 (0.63) PARP11PARP10KDM4EGRM5
SCHEMBL18500475 0.67 PARP10 (0.58) PARP11PARP10GRM5
SCHEMBL19441071 0.67 TDP1 (0.59) KDM4EMAPTSCN10A
SCHEMBL19308817 0.66 KDM4E (0.37) KDM4EMAPTSCN10A
SCHEMBL17461356 0.65 TDP1 (0.57) KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11806335-B2 Heterocyclic carboxylate compounds as glycolate oxidase inhibitors Lilac Therapeutics, Inc. (US) 2023-11-07 US disclosed
US-20210128532-A1 HETEROCYCLIC CARBOXYLATE COMPOUNDS AS GLYCOLATE OXIDASE INHIBITORS Lilac Therapeutics, Inc. 2021-05-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11806335-B2 Heterocyclic carboxylate compounds as glycolate oxidase inhibitors UGDH, PGD, PNPO PARP11 2694/4885PARP10 2086/4885KDM4E 1855/4885
US-20210128532-A1 HETEROCYCLIC CARBOXYLATE COMPOUNDS AS GLYCOLATE OXIDASE INHIBITORS UGDH, PGD, PNPO PARP11 2694/4885PARP10 2086/4885KDM4E 1855/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.