SCHEMBL23332016

SCHEMBL23332016

C=C(CC(=O)Oc1ccc(CC(NC(=O)OC(C)(C)C)C(=O)NC(C)(C)C(C)(C)C)cc1)C(=O)OC

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSS P25774 8/20 0.45
CTSK P43235 7/20 0.45
CTSB P07858 2/20 0.44
CTSL P07711 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
ITGB3 P05106 1/20 0.43
ITGA2B P08514 1/20 0.43
BCL2 P10415 1/20 0.42
REN P00797 4/20 0.41
ABCB1 P08183 1/20 0.40
AKT1 P31749 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23332002 0.92 CTSS (0.45) CTSSCTSKCTSBCTSLHDAC8
SCHEMBL24941612 0.89 CTSS (0.43) CTSSCTSKCTSBCTSLHDAC8
SCHEMBL24942215 0.83 CTSS (0.43) CTSSCTSKCTSBCTSLHDAC8
SCHEMBL23332014 0.82 CTSC (0.35) HDAC8
SCHEMBL23331990 0.81 CACNA1B (0.47) CTSSCTSKCTSBCTSLHDAC8
SCHEMBL24942213 0.81 CTSS (0.43) CTSSCTSKCTSBCTSLHDAC8
SCHEMBL23306678 0.81 CACNA1B (0.47) CTSSCTSKCTSBCTSLHDAC8
SCHEMBL23332134 0.79 CTSS (0.51) CTSSCTSKCTSBCTSLHDAC8
SCHEMBL23306474 0.78 REN (0.41) CTSSCTSKITGB3ITGA2BREN
SCHEMBL23306472 0.78 REN (0.41) CTSSCTSKITGB3ITGA2BREN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021087082-A1 PRODRUGS OF ITACONATE AND METHYL ITACONATE THE JOHNS HOPKINS UNIVERSITY (US) 2021-05-06 WO disclosed
WO-2021087083-A1 USE OF ITACONATE AND ITS DERIVATIVES/ANALOGUES TO INDUCE HAIR GROWTH THE JOHNS HOPKINS UNIVERSITY (US) 2021-05-06 WO disclosed