SCHEMBL23331990

SCHEMBL23331990

C=C(CC(=O)Oc1ccc(C[C@H](NC(=O)OC(C)(C)C)C(=O)OCc2ccccc2)cc1)C(=O)OC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 1/20 0.47
KLK5 Q9Y337 1/20 0.47
CTSS P25774 3/20 0.47
CTSK P43235 2/20 0.47
CTSL P07711 1/20 0.47
CTSB P07858 1/20 0.47
BCL2 P10415 1/20 0.47
REN P00797 1/20 0.46
PPARA Q07869 1/20 0.46
ACE P12821 1/20 0.46
PTPN1 P18031 1/20 0.45
ITGB3 P05106 1/20 0.45
ITGA2B P08514 1/20 0.45
EPHX2 P34913 1/20 0.45
ABCB1 P08183 1/20 0.45
MAPT P10636 2/20 0.44
HDAC8 Q9BY41 1/20 0.44
KDM4E B2RXH2 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
POLB P06746 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23306678 1.00 CACNA1B (0.47) CACNA1BKLK5CTSSCTSKCTSL
SCHEMBL23306289 0.93 REN (0.48) CACNA1BKLK5CTSSCTSKCTSL
SCHEMBL23332228 0.93 REN (0.48) CACNA1BKLK5CTSSCTSKCTSL
SCHEMBL23331991 0.84 PPARA (0.50) KLK5CTSSCTSKCTSLCTSB
SCHEMBL6780588 0.84 CTSS (0.54) KLK5CTSSCTSKCTSLCTSB
SCHEMBL24925616 0.84 KLK5 (0.52) CACNA1BKLK5CTSSCTSKCTSL
SCHEMBL6438287 0.84 CACNA1B (0.60) CACNA1BKLK5CTSSCTSKCTSL
SCHEMBL7292396 0.84 CACNA1B (0.60) CACNA1BKLK5CTSSCTSKCTSL
SCHEMBL9240969 0.84 CACNA1B (0.60) CACNA1BKLK5CTSSCTSKCTSL
SCHEMBL22404737 0.83 CTSS (0.64) KLK5CTSSCTSKCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230028516-A1 PRODRUGS OF ITACONATE AND METHYL ITACONATE INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY AS CR V.V.I. (CZ) 2023-01-26 US disclosed
WO-2021087082-A1 PRODRUGS OF ITACONATE AND METHYL ITACONATE THE JOHNS HOPKINS UNIVERSITY (US) 2021-05-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230028516-A1 PRODRUGS OF ITACONATE AND METHYL ITACONATE HADHA, IMPDH1, CYP27A1 CACNA1B 4707/4885KLK5 2976/4885CTSS 1933/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.