SCHEMBL23337429

SCHEMBL23337429

CN1CCc2[nH]cnc2C1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
BLM P54132 1/20 0.40
HTR1A P08908 2/20 0.39
DRD2 P14416 2/20 0.39
HTR2A P28223 2/20 0.39
BUB1 O43683 2/20 0.37
PDE5A O76074 1/20 0.34
MAPK1 P28482 1/20 0.33
NEK2 P51955 1/20 0.32
ATAD2 Q6PL18 1/20 0.32
ADORA2B P29275 3/20 0.31
ADORA2A P29274 2/20 0.31
ALDH1A1 P00352 1/20 0.31
PIK3CD O00329 1/20 0.31
ALPL P05186 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
TMIGD3 P0DMS9 1/20 0.31
PDE4A P27815 1/20 0.31
ADORA1 P30542 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11923830 0.81 MEN1 (0.42) MEN1KMT2ABLMHTR1ADRD2
SCHEMBL23336559 0.78 HTR1A (0.35) MEN1KMT2ABLMHTR1ADRD2
SCHEMBL5793769 0.69
SCHEMBL5138845 0.66 KMT2A (0.41) MEN1KMT2ABLMHTR1ADRD2
SCHEMBL16188711 0.64 MEN1 (0.36) MEN1KMT2ABUB1ATAD2GRM5
SCHEMBL23337430 0.64 ALDH1A1 (0.43) MEN1KMT2AHTR1ADRD2HTR2A
SCHEMBL30969607 0.64 CDC7 (0.43) MAPK1
SCHEMBL12082637 0.64 AKT1 (0.39) DRD2CYP2C19
SCHEMBL16626803 0.63 GRM5 (0.33) MEN1KMT2AALDH1A1GRM5
SCHEMBL2669115 0.63 GRM5 (0.39) MEN1KMT2AGRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021133894-A1 BTK INHIBITORS BIOGEN MA INC. (US) 2021-07-01 WO disclosed
WO-2021087086-A1 CONDENSED PYRIDAZINE OR PYRIMIDINE AS BTK INHIBITORS BIOGEN MA INC. (US) 2021-05-06 WO disclosed