SCHEMBL23342005

SCHEMBL23342005

CSC(=O)N1CCN(C(=O)N(C)C(C)C)CC1

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.34
ALDH1A1 P00352 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
GRM5 P41594 1/20 0.33
HTR1A P08908 1/20 0.32
KMT2A Q03164 2/20 0.31
MEN1 O00255 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12807825 0.78
SCHEMBL12872504 0.78 HTR1A (0.53) MAPTALDH1A1HTR1A
SCHEMBL25912762 0.77 L3MBTL1 (0.33) MAPTL3MBTL1SMN1; SMN2
SCHEMBL14319076 0.77 SMN1; SMN2 (0.39) MAPTALDH1A1KMT2AMEN1SMN1; SMN2
SCHEMBL20346243 0.76 HRH3 (0.44) MAPT
SCHEMBL25895293 0.76 CHRNB2 (0.38) MAPTALDH1A1HTR1AKMT2AMEN1
SCHEMBL21733089 0.76 MAPT (0.33) MAPTHTR1AKMT2AMEN1SMN1; SMN2
SCHEMBL20234147 0.74 HRH3 (0.44) MAPTALDH1A1
SCHEMBL22152624 0.73 KDM4E (0.44) ALDH1A1HTR1A
SCHEMBL18705032 0.73 HRH3 (0.36) MAPTALDH1A1L3MBTL1GRM5HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11739074-B2 Ras inhibitors Revolution Medicines, Inc. (US) 2023-08-29 US disclosed
US-20210130326-A1 RAS INHIBITORS WILMINGTON TRUST, NATIONAL ASSOCIATION, AS AGENT 2021-05-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11739074-B2 Ras inhibitors KRAS, NRAS, HRAS MAPT 3764/4885ALDH1A1 3951/4885L3MBTL1 3587/4885
US-20210130326-A1 RAS INHIBITORS KRAS, NRAS, HRAS MAPT 3364/4885ALDH1A1 4437/4885L3MBTL1 3097/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.