SCHEMBL23355180

SCHEMBL23355180

Cc1ccc(F)c(C(=O)NC(C=O)Cc2ccccc2)c1Cl

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 11/20 0.49
L3MBTL1 Q9Y468 1/20 0.43
CTSB P07858 2/20 0.43
ITGB1 P05556 1/20 0.41
ITGA4 P13612 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24008805 0.85 CAPN1 (0.52) CAPN1CTSB
SCHEMBL23355177 0.82 CAPN1 (0.58) CAPN1CTSBITGA4
SCHEMBL29961792 0.81 CAPN1 (0.58) CAPN1L3MBTL1ITGB1ITGA4
SCHEMBL24008799 0.81 CAPN1 (0.58) CAPN1L3MBTL1ITGB1ITGA4
SCHEMBL28558990 0.79 L3MBTL1 (0.41) CAPN1L3MBTL1ITGB1ITGA4
SCHEMBL23355169 0.77 CAPN1 (0.58) CAPN1CTSBITGB1ITGA4
SCHEMBL23355192 0.75 ITGA4 (0.56) CAPN1ITGB1ITGA4
SCHEMBL24862871 0.75 CAPN1 (0.73) CAPN1CTSB
SCHEMBL24862869 0.75 CAPN1 (0.69) CAPN1CTSB
SCHEMBL24008869 0.74 CAPN1 (0.48) CAPN1CTSBITGB1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220347173-A1 METHODS OF TREATING LIVER FIBROSIS USING CALPAIN INHIBITORS BLADE THERAPEUTICS INC (US) 2022-11-03 US disclosed
US-20210347727-A1 CALPAIN MODULATORS AND THERAPEUTIC USES THEREOF BLADE THERAPEUTICS, INC. 2021-11-11 US disclosed
EP-3820864-A1 METHODS OF TREATING LIVER FIBROSIS USING CALPAIN INHIBITORS Blade Therapeutics, Inc. (US) 2021-05-19 EP disclosed
CN-112703188-A Method for treating liver fibrosis using calpain inhibitor 布莱德治疗公司 2021-04-23 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210347727-A1 CALPAIN MODULATORS AND THERAPEUTIC USES THEREOF CAPN1, CAPNS1, CAPN2 CAPN1 1/4885L3MBTL1 2837/4885CTSB 56/4885
US-20220347173-A1 METHODS OF TREATING LIVER FIBROSIS USING CALPAIN INHIBITORS CAPNS1, CAPN9, CAPN2 CAPN1 4/4885L3MBTL1 3900/4885CTSB 24/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.