SCHEMBL23355378

SCHEMBL23355378

O=C(O)Nc1ccc(Oc2nc(Br)cs2)cc1F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.37
KDR P35968 3/20 0.37
MET P08581 1/20 0.37
SMN1; SMN2 Q16637 3/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
MAPT P10636 1/20 0.36
MAPK1 P28482 1/20 0.36
RECQL P46063 1/20 0.36
NPC1 O15118 3/20 0.35
RAB9A P51151 3/20 0.35
ALDH1A1 P00352 2/20 0.35
GAA P10253 2/20 0.35
HPGD P15428 1/20 0.35
ALOX12 P18054 1/20 0.35
CASP3 P42574 1/20 0.35
SENP7 Q9BQF6 1/20 0.35
SENP6 Q9GZR1 1/20 0.35
ABL1 P00519 1/20 0.35
GCK P35557 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29834682 0.84 CYP17A1 (0.43) KDRABL1
SCHEMBL23368116 0.84 CYP17A1 (0.43) KDRABL1
SCHEMBL23355406 0.80 SCN9A (0.36) LMNAKDRMETSMN1; SMN2MEN1
SCHEMBL23355335 0.79 LMNA (0.41) LMNAKDRMETSMN1; SMN2RAB9A
SCHEMBL23355472 0.79 CA1 (0.35) LMNAKDRMETABL1GCK
SCHEMBL23355401 0.77 MEN1 (0.41) LMNAKDRSMN1; SMN2MEN1KMT2A
SCHEMBL24037369 0.75 ALDH1A1 (0.34) ALDH1A1GCK
SCHEMBL23355350 0.74 MAPK14 (0.35) KDRMETSMN1; SMN2MEN1KMT2A
SCHEMBL23355301 0.73 NPC1 (0.48) LMNASMN1; SMN2MEN1KMT2AMAPT
SCHEMBL21612809 0.72 CYP17A1 (0.42) LMNAKDRABL1KITPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230025510-A1 BIARYL ETHER-TYPE QUINAZOLINE DERIVATIVES DAIICHI SANKYO COMPANY, LIMITED (JP) 2023-01-26 US disclosed
EP-3822263-A1 BIARYL ETHER-TYPE QUINAZOLINE DERIVATIVE Daiichi Sankyo Company, Limited (JP) 2021-05-19 EP disclosed
CN-112334460-A Biaryl ether type quinazoline derivative 第一三共株式会社 2021-02-05 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230025510-A1 BIARYL ETHER-TYPE QUINAZOLINE DERIVATIVES ERBB2, EGFR, ERBB3 LMNA 4004/4885KDR 20/4885MET 34/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.