SCHEMBL23355459

SCHEMBL23355459

CC(C)(C)N(C(=O)O)c1ccc(Oc2cccc(C(=O)NN)c2)cc1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
LMNA P02545 2/20 0.42
HDAC8 Q9BY41 1/20 0.42
NPC1 O15118 4/20 0.41
RAB9A P51151 4/20 0.41
POLB P06746 1/20 0.41
CYP2C9 P11712 1/20 0.41
KDM4E B2RXH2 2/20 0.39
GCK P35557 1/20 0.38
TNKS O95271 1/20 0.38
PARP15 Q460N3 1/20 0.38
PARP14 Q460N5 1/20 0.38
PARP10 Q53GL7 1/20 0.38
TNKS2 Q9H2K2 1/20 0.38
PARP2 Q9UGN5 1/20 0.38
ERCC5 P28715 1/20 0.38
FEN1 P39748 1/20 0.38
PKM P14618 1/20 0.37
AKR1C3 P42330 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28909804 0.88 KMO (0.47) ALDH1A1SMN1; SMN2LMNAHDAC8NPC1
SCHEMBL23355435 0.75 RAB9A (0.51) SMN1; SMN2LMNAHDAC8NPC1RAB9A
SCHEMBL28538655 0.74 KDM4E (0.37) ALDH1A1SMN1; SMN2LMNANPC1RAB9A
SCHEMBL2830822 0.74 HDAC8 (0.73) ALDH1A1SMN1; SMN2LMNAHDAC8NPC1
SCHEMBL31295303 0.74 HDAC8 (0.73) ALDH1A1SMN1; SMN2LMNAHDAC8NPC1
SCHEMBL23355461 0.74 RAB9A (0.48) SMN1; SMN2LMNANPC1RAB9APOLB
SCHEMBL2649884 0.74 FABP1 (0.57) ALDH1A1SMN1; SMN2LMNAHDAC8NPC1
SCHEMBL519443 0.72 MAPT (0.37) ALDH1A1SMN1; SMN2LMNAPOLBCYP2C9
SCHEMBL519129 0.72 FFAR4 (0.39)
SCHEMBL7229522 0.72 NPC1 (0.64) ALDH1A1SMN1; SMN2LMNAHDAC8NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3822263-A1 BIARYL ETHER-TYPE QUINAZOLINE DERIVATIVE Daiichi Sankyo Company, Limited (JP) 2021-05-19 EP disclosed
CN-112334460-A Biaryl ether type quinazoline derivative 第一三共株式会社 2021-02-05 CN disclosed