SCHEMBL23355470

SCHEMBL23355470

COc1cc2nc(-c3ccc(Oc4cccc(-c5nnc(C(C)C)o5)c4)cc3F)nc(N)c2cc1N

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.36
KMT2A Q03164 3/20 0.36
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CA9 Q16790 2/20 0.34
CA13 Q8N1Q1 2/20 0.34
TP53 P04637 5/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
NPC1 O15118 3/20 0.33
RAB9A P51151 3/20 0.33
MAPT P10636 3/20 0.33
HPGD P15428 2/20 0.33
MEN1 O00255 2/20 0.33
ALDH1A1 P00352 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PIM1 P11309 1/20 0.33
PIM3 Q86V86 1/20 0.33
PIM2 Q9P1W9 1/20 0.33
POLB P06746 2/20 0.33
ATR Q13535 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23355338 0.90 KDM4E (0.38) KDM4EKMT2ACA1CA2CA9
SCHEMBL23355389 0.87 KDM4E (0.36) KDM4EKMT2ACA1CA2CA9
SCHEMBL23355422 0.80 ADORA1 (0.34) KDM4EKMT2ATP53SMN1; SMN2MAPT
SCHEMBL23355413 0.78 LRRK2 (0.40) KDM4ETP53SMN1; SMN2NPC1RAB9A
SCHEMBL23368182 0.78 EGFR (0.47)
SCHEMBL23368158 0.77 KDM4E (0.45) KDM4EKMT2ATP53SMN1; SMN2NPC1
SCHEMBL23355355 0.70 LRRK2 (0.32)
SCHEMBL15877172 0.70 SLC2A1 (0.43) KDM4EKMT2ATP53NPC1MAPT
Trifluoroacetic Acid SCHEMBL23355453 0.70 SMN1; SMN2 (0.39) KDM4EKMT2ATP53SMN1; SMN2NPC1
SCHEMBL23355331 0.69 MAPT (0.40) KDM4EKMT2ACA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3822263-A1 BIARYL ETHER-TYPE QUINAZOLINE DERIVATIVE Daiichi Sankyo Company, Limited (JP) 2021-05-19 EP disclosed