SCHEMBL2335862

SCHEMBL2335862

COc1c[c]c([N+](=O)[O-])cc1OCCCBr

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 9/20 0.37
SMN1; SMN2 Q16637 5/20 0.37
HPGD P15428 5/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
LMNA P02545 5/20 0.36
ALDH1A1 P00352 6/20 0.35
MAPK1 P28482 1/20 0.35
HTT P42858 2/20 0.35
GAA P10253 1/20 0.33
S1PR4 O95977 1/20 0.33
KMT2A Q03164 1/20 0.33
CTSB P07858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3392935 0.96 MAPT (0.37) MAPTSMN1; SMN2HPGDNPC1RAB9A
SCHEMBL3392298 0.95 MAPT (0.36) MAPTSMN1; SMN2HPGDNPC1RAB9A
SCHEMBL123690 0.82 ALDH1A1 (0.43) MAPTSMN1; SMN2NPC1CYP3A4CYP2D6
SCHEMBL10527285 0.78 CYP19A1 (0.42) MAPTSMN1; SMN2NPC1RAB9ALMNA
SCHEMBL28401883 0.78 KDM4E (0.39) MAPTHPGDCYP1A2CYP3A4CYP2D6
SCHEMBL13673810 0.76 MEN1 (0.47) MAPTSMN1; SMN2HPGDNPC1RAB9A
SCHEMBL6927577 0.74 MAPT (0.60) MAPTSMN1; SMN2HPGDNPC1RAB9A
SCHEMBL28738082 0.74 HTT (0.38) MAPTCYP3A4ALDH1A1HTTKMT2A
SCHEMBL21808035 0.74 HTT (0.38) MAPTSMN1; SMN2CYP3A4LMNAALDH1A1
SCHEMBL1356676 0.74 ALDH1A1 (0.47) MAPTSMN1; SMN2CYP3A4LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2358719-B1 Novel pyrrolo[2,1-c][1,4]benzodiazepine derivatives with dithiocarbamate side chains and process for the preparation thereof COUNCIL SCIENT IND RES (IN) 2014-10-01 EP disclosed
EP-2358719-A1 Novel pyrroiol2,l-cu1.41benzodiazepine derivatives with dithiocarbamate side chains and process for the preparation thereof Council Of Scientific & Industrial Research (IN) 2011-08-24 EP disclosed
WO-2010058414-A1 NOVEL PYRROIOL2,L-CU1.41BENZODIAZEPINE DERIVATIVES WITH DITHIOCARBAMATE SIDE CHAINS AND PROCESS FOR THE PREPARATION THEREOF COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2010-05-27 WO disclosed