SCHEMBL23364207

SCHEMBL23364207

CC(C)(C)[Si](C)(C)OCC[C@H]1CCC(=O)N1

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DUT P33316 2/20 0.35
CD274 Q9NZQ7 3/20 0.32
PDCD1LG2 Q9BQ51 2/20 0.32
IRAK4 Q9NWZ3 1/20 0.32
PDCD1 Q15116 1/20 0.31
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23363973 1.00 DUT (0.35) DUTCD274PDCD1LG2IRAK4PDCD1
SCHEMBL16447361 1.00 DUT (0.35) DUTCD274PDCD1LG2IRAK4PDCD1
SCHEMBL211169 0.84 IRAK4 (0.37) DUTIRAK4
SCHEMBL964133 0.84 IRAK4 (0.37) DUTIRAK4
SCHEMBL211911 0.84 IRAK4 (0.37) DUTIRAK4
SCHEMBL26481101 0.79 DUT (0.34) DUT
SCHEMBL29231913 0.79 DUT (0.34) DUT
SCHEMBL24335316 0.78 IRAK4 (0.34) CD274PDCD1LG2IRAK4PDCD1LMNA
SCHEMBL4988554 0.77 CD274 (0.32) CD274PDCD1LG2IRAK4PDCD1LMNA
SCHEMBL21802067 0.76 IRAK4 (0.36) DUTCD274PDCD1LG2IRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230002383-A1 NOVEL FUNCTIONALIZED LACTAMS AS MODULATORS OF THE 5-HYDROXYTRYPTAMINE RECEPTOR 7 AND THEIR METHOD OF USE PRAEVENTIX, LLC 2023-01-05 US disclosed
US-20230002383-A1 NOVEL FUNCTIONALIZED LACTAMS AS MODULATORS OF THE 5-HYDROXYTRYPTAMINE RECEPTOR 7 AND THEIR METHOD OF USE PRAEVENTIX, LLC 2023-01-05 US disclosed
EP-4058455-A1 NOVEL FUNCTIONALIZED LACTAMS AS MODULATORS OF THE 5-HYDROXYTRYPTAMINE RECEPTOR 7 AND THEIR METHOD OF USE Temple University - Of The Commonwealth System of Higher Education (US) 2022-09-21 EP disclosed
CN-115003675-A Novel functionalized lactams as 5-hydroxytryptamine receptor 7 modulators and methods of use thereof 英联邦高等教育系统坦普尔大学 2022-09-02 CN disclosed
WO-2021097116-A1 NOVEL FUNCTIONALIZED LACTAMS AS MODULATORS OF THE 5-HYDROXYTRYPTAMINE RECEPTOR 7 AND THEIR METHOD OF USE TEMPLE UNIVERSITY-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2021-05-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230002383-A1 NOVEL FUNCTIONALIZED LACTAMS AS MODULATORS OF THE 5-HYDROXYTRYPTAMINE RECEPTOR 7 AND THEIR METHOD OF USE HTR7, HTR1A, HTR2C DUT 2029/4885CD274 3908/4885PDCD1LG2 3250/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.