SCHEMBL2337016

SCHEMBL2337016

CC(C)OC1CCC(Cl)(c2ccc3c(c2)CN(C(=O)OC(C)(C)C)Cc2nncn2-3)CC1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 2/20 0.35
CRBN Q96SW2 2/20 0.35
OXTR P30559 3/20 0.35
AVPR1A P37288 1/20 0.35
IDH1 O75874 2/20 0.33
ESR2 Q92731 1/20 0.32
GPR119 Q8TDV5 2/20 0.32
MAP3K5 Q99683 2/20 0.31
NR1H2 P55055 2/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31
CTSD P07339 1/20 0.31
CTSE P14091 1/20 0.31
BACE1 P56817 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2340822 0.90 DDB1 (0.37) DDB1CRBNOXTRAVPR1AIDH1
SCHEMBL2336887 0.89 PDE4B (0.36) DDB1CRBNOXTRAVPR1AESR2
SCHEMBL2341708 0.89 DDB1 (0.34) DDB1CRBNOXTRAVPR1AESR2
SCHEMBL2340272 0.89 DDB1 (0.35) DDB1CRBNOXTRAVPR1AESR2
SCHEMBL2336519 0.89 DDB1 (0.35) DDB1CRBNOXTRAVPR1AESR2
SCHEMBL2469674 0.87 PDE4A (0.34) DDB1CRBNOXTRAVPR1AESR2
SCHEMBL2550063 0.86 NAMPT (0.40) DDB1CRBNOXTRAVPR1AESR2
SCHEMBL2469541 0.85 GPR119 (0.34) DDB1CRBNOXTRAVPR1AESR2
SCHEMBL2573980 0.85 DDB1 (0.38) DDB1CRBNOXTRAVPR1AESR2
SCHEMBL2579657 0.85 OXTR (0.36) DDB1CRBNOXTRAVPR1AESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2358714-A1 ALKYLCYCLOHEXYLETHERS OF DIHYDROTETRAAZABENZOAZULENES F. Hoffmann-La Roche AG (CH) 2011-08-24 EP claimed
WO-2010057795-A1 ALKYLCYCLOHEXYLETHERS OF DIHYDROTETRAAZABENZOAZULENES F. HOFFMANN-LA ROCHE AG (CH) 2010-05-27 WO claimed
EP-2358714-A1 ALKYLCYCLOHEXYLETHERS OF DIHYDROTETRAAZABENZOAZULENES F. Hoffmann-La Roche AG (CH) 2011-08-24 EP disclosed
WO-2010057795-A1 ALKYLCYCLOHEXYLETHERS OF DIHYDROTETRAAZABENZOAZULENES F. HOFFMANN-LA ROCHE AG (CH) 2010-05-27 WO disclosed