SCHEMBL2337751

SCHEMBL2337751

COc1ccc(C2C(C(=O)Nc3cccc(OC)c3)c3cc(OC)c(OC)cc3C(=O)N2C)cc1.COc1cccc(NC(=O)C2c3cc(OC)c(OC)cc3C(=O)N(C)C2c2ccc(OC)c(OC)c2)c1

nearest known ligand 0.74

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.74
CYP3A4 P08684 3/20 0.73
ALOX15 P16050 3/20 0.66
TSHR P16473 3/20 0.66
KMT2A Q03164 3/20 0.63
CYP2C9 P11712 2/20 0.63
MEN1 O00255 1/20 0.63
NPC1 O15118 1/20 0.61
ALDH1A1 P00352 3/20 0.59
HTT P42858 2/20 0.59
MAPK1 P28482 1/20 0.58
NPSR1 Q6W5P4 1/20 0.57
LMNA P02545 2/20 0.57
MDM2 Q00987 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
HSD17B10 Q99714 3/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
MAPT P10636 1/20 0.54
POLB P06746 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2332683 0.97 CYP3A4 (0.76) GAACYP3A4ALOX15TSHRKMT2A
SCHEMBL2335153 0.96 GAA (0.79) GAACYP3A4ALOX15TSHRKMT2A
SCHEMBL2334030 0.89 GAA (0.82) GAACYP3A4ALOX15TSHRKMT2A
SCHEMBL2336448 0.85 GAA (1.00) GAACYP3A4TSHRNPC1ALDH1A1
SCHEMBL2340254 0.83 CYP3A4 (0.69) GAACYP3A4ALOX15TSHRKMT2A
SCHEMBL2334861 0.82 CYP3A4 (0.68) GAACYP3A4ALOX15TSHRKMT2A
SCHEMBL2334417 0.74 GAA (0.59) GAACYP3A4TSHRKMT2ACYP2C9
SCHEMBL2339357 0.74 CYP3A4 (0.57) GAACYP3A4KMT2ACYP2C9MEN1
SCHEMBL2330482 0.73 GAA (0.77) GAACYP3A4TSHRKMT2AMEN1
SCHEMBL252628 0.73 CYP3A4 (0.79) GAACYP3A4ALOX15TSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2358682-A2 ISOQUINOLONE DERIVATIVES AS INHIBITORS OF PLAVIVIRUS REPLICATION Katholieke Universiteit Leuven, K.U. Leuven R&D (BE) 2011-08-24 EP disclosed