SCHEMBL2335153

SCHEMBL2335153

COc1ccc(C2C(C(=O)Nc3cccc(OC)c3)c3cc(OC)c(OC)cc3C(=O)N2C)cc1

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.79
CYP3A4 P08684 4/20 0.77
NPC1 O15118 1/20 0.65
CYP2C9 P11712 4/20 0.62
KMT2A Q03164 3/20 0.62
MEN1 O00255 1/20 0.62
MAPK1 P28482 1/20 0.62
ALOX15 P16050 4/20 0.61
HTT P42858 2/20 0.61
NPSR1 Q6W5P4 1/20 0.61
LMNA P02545 1/20 0.60
MDM2 Q00987 1/20 0.60
L3MBTL1 Q9Y468 1/20 0.60
TSHR P16473 3/20 0.60
SMN1; SMN2 Q16637 1/20 0.59
ALDH1A1 P00352 4/20 0.58
KDM4E B2RXH2 1/20 0.54
MAPT P10636 1/20 0.54
CYP1A2 P05177 2/20 0.54
CYP2C19 P33261 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2337751 0.96 GAA (0.74) GAACYP3A4NPC1CYP2C9KMT2A
SCHEMBL2332683 0.93 CYP3A4 (0.76) GAACYP3A4NPC1CYP2C9KMT2A
SCHEMBL2336448 0.88 GAA (1.00) GAACYP3A4NPC1LMNATSHR
SCHEMBL2340254 0.86 CYP3A4 (0.69) GAACYP3A4NPC1CYP2C9KMT2A
SCHEMBL2334861 0.85 CYP3A4 (0.68) GAACYP3A4NPC1CYP2C9KMT2A
SCHEMBL2334030 0.85 GAA (0.82) GAACYP3A4NPC1CYP2C9KMT2A
SCHEMBL2334417 0.77 GAA (0.59) GAACYP3A4NPC1CYP2C9KMT2A
SCHEMBL2339357 0.76 CYP3A4 (0.57) GAACYP3A4NPC1CYP2C9KMT2A
SCHEMBL2330482 0.76 GAA (0.77) GAACYP3A4NPC1KMT2AMEN1
SCHEMBL252628 0.76 CYP3A4 (0.79) GAACYP3A4NPC1CYP2C9KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110224208-A1 NOVEL INHIBITORS OF FLAVIVIRUS REPLICATION KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2011-09-15 US claimed
EP-2358682-A2 ISOQUINOLONE DERIVATIVES AS INHIBITORS OF PLAVIVIRUS REPLICATION Katholieke Universiteit Leuven, K.U. Leuven R&D (BE) 2011-08-24 EP claimed
WO-2010055164-A2 NOVEL INHIBITORS OF FLAVIVIRUS REPLICATION KATHOLIEKE UNIVERSITEIT LEUVEN, K.U.LEUVEN R&D (BE) 2010-05-20 WO claimed
US-20110224208-A1 NOVEL INHIBITORS OF FLAVIVIRUS REPLICATION KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2011-09-15 US disclosed
EP-2358682-A2 ISOQUINOLONE DERIVATIVES AS INHIBITORS OF PLAVIVIRUS REPLICATION Katholieke Universiteit Leuven, K.U. Leuven R&D (BE) 2011-08-24 EP disclosed
WO-2010055164-A2 NOVEL INHIBITORS OF FLAVIVIRUS REPLICATION KATHOLIEKE UNIVERSITEIT LEUVEN, K.U.LEUVEN R&D (BE) 2010-05-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110224208-A1 NOVEL INHIBITORS OF FLAVIVIRUS REPLICATION MAVS, IRF3, EIF2AK2 GAA 2348/4885CYP3A4 722/4885NPC1 858/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.