SCHEMBL2340091

SCHEMBL2340091

O=C(Nc1nnc(-c2cccc(Cl)c2)o1)N1CCC2(CC1)CC(c1cccc(OC(F)(F)F)c1)C2

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 5/20 0.50
USP30 Q70CQ3 1/20 0.42
TRPM8 Q7Z2W7 5/20 0.39
TRPV1 Q8NER1 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.38
MEN1 O00255 1/20 0.38
HPGD P15428 1/20 0.38
MAPK1 P28482 1/20 0.38
CCR6 P51684 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KDM4E B2RXH2 3/20 0.37
EPHX2 P34913 2/20 0.37
ALDH1A1 P00352 1/20 0.37
P2RY14 Q15391 1/20 0.37
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2340079 0.85 MGLL (0.55) MGLLTRPM8TRPV1EPHX2
SCHEMBL2344291 0.77 MGLL (0.51) MGLLEPHX2
SCHEMBL22594321 0.75 KDM4E (0.61) L3MBTL1MEN1HPGDMAPK1CCR6
SCHEMBL2341031 0.74 MGLL (0.52) MGLLTRPM8TRPV1EPHX2ALDH1A1
SCHEMBL2422288 0.74 MGLL (0.61) MGLLTRPM8TRPV1EPHX2
SCHEMBL23859715 0.74 MGLL (0.63) MGLLEPHX2
SCHEMBL2341810 0.74 MGLL (0.49) MGLLTRPM8TRPV1EPHX2
SCHEMBL2347224 0.72 MGLL (0.50) MGLLTRPM8TRPV1EPHX2POLB
SCHEMBL29470023 0.70 MGLL (0.58) MGLL
SCHEMBL23868006 0.70 MGLL (0.58) MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2358704-A1 7-azaspiro [3.5]nonane-7-carboxamide compounds as modulators of fatty acid amide hydrolase Pfizer Inc. (US) 2011-08-24 EP claimed
US-20100113465-A1 7-AZASPIRO[3.5]NONANE-7-CARBOXAMIDE COMPOUNDS PFIZER INC. 2010-05-06 US claimed
WO-2010049841-A1 7-AZASPIRO [3.5] NONANE-7-CARBOXAMIDE COMPOUNDS AS MODULATORS OF FATTY ACID AMIDE HYDROLASE PFIZER INC. (US) 2010-05-06 WO claimed
US-20100113465-A1 7-AZASPIRO[3.5]NONANE-7-CARBOXAMIDE COMPOUNDS PFIZER INC. 2010-05-06 US disclosed
US-20100113465-A1 7-AZASPIRO[3.5]NONANE-7-CARBOXAMIDE COMPOUNDS PFIZER INC. 2010-05-06 US disclosed
US-20100113465-A1 7-AZASPIRO[3.5]NONANE-7-CARBOXAMIDE COMPOUNDS PFIZER INC. 2010-05-06 US disclosed
WO-2010049841-A1 7-AZASPIRO [3.5] NONANE-7-CARBOXAMIDE COMPOUNDS AS MODULATORS OF FATTY ACID AMIDE HYDROLASE PFIZER INC. (US) 2010-05-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100113465-A1 7-AZASPIRO[3.5]NONANE-7-CARBOXAMIDE COMPOUNDS FAAH, FAAH2, APEH MGLL 298/4885USP30 1217/4885TRPM8 1517/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.