SCHEMBL2340431

SCHEMBL2340431

O=C1CCCCN1c1cc[c]nc1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
AKR1C3 P42330 6/20 0.40
HPGD P15428 4/20 0.40
BRD9 Q9H8M2 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HRH3 Q9Y5N1 3/20 0.37
GAA P10253 2/20 0.35
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2342728 0.98 HPGD (0.42) ALDH1A1AKR1C3HPGDBRD9CYP1A2
SCHEMBL2337506 0.95 ALDH1A1 (0.46) ALDH1A1AKR1C3HPGDCYP1A2CYP3A4
SCHEMBL2347313 0.80 ALDH1A1 (0.38) ALDH1A1HPGD
SCHEMBL2350173 0.80 HPGD (0.38) AKR1C3HPGDGAA
SCHEMBL182890 0.78 ALDH1A1 (0.51) ALDH1A1AKR1C3HPGDBRD9CYP1A2
SCHEMBL23387936 0.75 MEN1 (0.31) ALDH1A1
SCHEMBL2342841 0.75 SLC6A2 (0.40) HPGD
SCHEMBL16570287 0.75 SLC6A2 (0.40)
SCHEMBL2344200 0.75 PTGS2 (0.44)
SCHEMBL255160 0.74 AKR1C3 (0.51) ALDH1A1AKR1C3HPGDBRD9HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115003663-B Novel heteroaryl-triazole compounds as pesticides 拜耳公司 2024-04-30 CN claimed
US-20230058623-A1 NOVEL HETEROARYL-TRIAZOLE COMPOUNDS AS PESTICIDES ELANCO ANIMAL HEALTH GMBH (DE) 2023-02-23 US claimed
CN-115003663-A Novel heteroaryl-triazole compounds as pesticides 拜耳公司 2022-09-02 CN claimed
WO-2021099303-A1 NOVEL HETEROARYL-TRIAZOLE COMPOUNDS AS PESTICIDES BAYER AKTIENGESELLSCHAFT (DE) 2021-05-27 WO claimed
CN-115003663-B Novel heteroaryl-triazole compounds as pesticides 拜耳公司 2024-04-30 CN disclosed
US-20230058623-A1 NOVEL HETEROARYL-TRIAZOLE COMPOUNDS AS PESTICIDES ELANCO ANIMAL HEALTH GMBH (DE) 2023-02-23 US disclosed
CN-115003663-A Novel heteroaryl-triazole compounds as pesticides 拜耳公司 2022-09-02 CN disclosed
WO-2021099303-A1 NOVEL HETEROARYL-TRIAZOLE COMPOUNDS AS PESTICIDES BAYER AKTIENGESELLSCHAFT (DE) 2021-05-27 WO disclosed
US-20110230467-A1 4,6-DIAMINONICOTINAMIDE COMPOUND ASTELLAS PHARMA INC. (JP) 2011-09-22 US disclosed
EP-2361902-A1 4,6-DIAMINONICOTINAMIDE COMPOUND Astellas Pharma Inc. (JP) 2011-08-31 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110230467-A1 4,6-DIAMINONICOTINAMIDE COMPOUND JAK3, JAK2, JAK1 ALDH1A1 1378/4885AKR1C3 2605/4885HPGD 2840/4885
US-20230058623-A1 NOVEL HETEROARYL-TRIAZOLE COMPOUNDS AS PESTICIDES PRXL2A, GLRX3, CYP4F3 ALDH1A1 4213/4885AKR1C3 894/4885HPGD 4450/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.