Ethylene

Ethylene

SCHEMBL2344022

C=C.CN(C)CCCN=C=N

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.52
CYP2D6 P10635 1/20 0.52
ALDH1A1 P00352 3/20 0.38
HRH4 Q9H3N8 2/20 0.38
TSHR P16473 1/20 0.38
HRH2 P25021 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
HSD17B10 Q99714 1/20 0.36
DNM1 Q05193 3/20 0.32
BACH1 O14867 1/20 0.30
MAFK O60675 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL301678 0.95
Carbimide SCHEMBL8927383 0.93 CYP1A2 (0.54) CYP1A2CYP2D6ALDH1A1HRH4TSHR
Hydrochloric Acid SCHEMBL248532 0.93 CYP1A2 (0.54) CYP1A2CYP2D6ALDH1A1HRH4TSHR
Ethane SCHEMBL8026831 0.93 CYP1A2 (0.54) CYP1A2CYP2D6ALDH1A1HRH4TSHR
Hydrochloric Acid SCHEMBL28296907 0.91 CYP1A2 (0.52) CYP1A2CYP2D6ALDH1A1HRH4TSHR
Iodomethane SCHEMBL7521844 0.91 CYP1A2 (0.52) CYP1A2CYP2D6ALDH1A1HRH4TSHR
Ethane SCHEMBL2545448 0.91 CYP1A2 (0.52) CYP1A2CYP2D6ALDH1A1HRH4TSHR
SCHEMBL27686663 0.89 CYP1A2 (0.50) CYP1A2CYP2D6ALDH1A1HRH4TSHR
SCHEMBL3095991 0.88 CYP1A2 (0.48) CYP1A2CYP2D6ALDH1A1HRH4TSHR
Ethyl Chloride SCHEMBL19668563 0.87 CYP1A2 (0.53) CYP1A2CYP2D6ALDH1A1HRH4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2679227-B1 NANOPARTICLE CONTAINING PROSTAGLANDIN I2 DERIVATIVE LTT BIO PHARMA CO LTD (JP) 2018-04-11 EP disclosed
EP-1985309-B1 NANOPARTICLES CONTAINING WATER-SOLUBLE NON-PEPTIDE LOW-MOLECULAR WEIGHT DRUG LTT BIO PHARMA CO LTD (JP) 2016-11-23 EP disclosed
US-9161986-B2 Nanoparticle containing prostaglandin I2 derivative LTT BIO-PHARMA CO., LTD. (JP) 2015-10-20 US disclosed
US-8916206-B2 Nanoparticles containing water-soluble non-peptide low-molecular weight drug LTT BIO-PHARMA CO., LTD. (JP) 2014-12-23 US disclosed
US-20140050690-A1 NANOPARTICLE CONTAINING PROSTAGLANDIN I 2 DERIVATIVE LTT BIO-PHARMA CO., LTD. (JP) 2014-02-20 US disclosed
US-20110262548-A1 NOVEL PROSTAGLANDIN E1 DERIVATIVE AND NANOPARTICLE HAVING THE SAME ENCAPSULATED THEREIN LTT BIO-PHARMA CO., LTD. (JP) 2011-10-27 US disclosed
EP-2361918-A1 NOVEL PROSTAGLANDIN E1 DERIVATIVE, AND NANOPARTICLE HAVING SAME ENCAPSULATED THEREIN LTT Bio-Pharma Co., Ltd. (JP) 2011-08-31 EP disclosed
US-20100129456-A1 SUSTAINED-RELEASE NANOPARTICLE CONTAINING LOW-MOLECULAR-WEIGHT DRUG WITH NEGATIVELY CHARGED GROUP LTT BIO-PHARMA CO., LTD. (JP) 2010-05-27 US disclosed
EP-2156848-A1 LOW-MOLECULE DRUG-CONTAINING NANOPARTICLE HAVING SUSTAINED RELEASE NEGATIVELY CHARGED GROUP LTT Bio-Pharma Co., Ltd. (JP) 2010-02-24 EP disclosed
US-20090317479-A1 NANOPARTICLES CONTAINING WATER-SOLUBLE NON-PEPTIDE LOW-MOLECULAR WEIGHT DRUG LTT BIO-PHARMA CO., LTD. (JP) 2009-12-24 US disclosed
EP-1985309-A1 NANOPARTICLE CONTAINING WATER-SOLUBLE NON-PEPTIDIC LOW MOLECULAR WEIGHT SUBSTANCE LTT Bio-Pharma Co., Ltd. (JP) 2008-10-29 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110262548-A1 NOVEL PROSTAGLANDIN E1 DERIVATIVE AND NANOPARTICLE HAVING THE SAME ENCAPSULATED THEREIN PTGER1, PTGS1, PTGES CYP1A2 938/4885CYP2D6 1148/4885ALDH1A1 62/4885
US-20140050690-A1 NANOPARTICLE CONTAINING PROSTAGLANDIN I 2 DERIVATIVE PTGIS, PTGS2, PTGS1 CYP1A2 1282/4885CYP2D6 2550/4885ALDH1A1 888/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.