SCHEMBL2344535

SCHEMBL2344535

CC(C)(C)OC(=O)N1CCC2(CC1)CC(c1cccc(OS(=O)(=O)C(F)(F)F)c1)C2

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.47
DRD1 P21728 2/20 0.47
DRD4 P21917 2/20 0.47
DRD5 P21918 2/20 0.47
DRD3 P35462 2/20 0.47
GPR119 Q8TDV5 9/20 0.47
MGLL Q99685 5/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29470023 0.87 MGLL (0.58) GPR119MGLL
SCHEMBL23868006 0.87 MGLL (0.58) GPR119MGLL
SCHEMBL2428771 0.86 MGLL (0.59) DRD2DRD1DRD4DRD5DRD3
SCHEMBL2424111 0.86 MGLL (0.59) DRD2DRD1DRD4DRD5DRD3
SCHEMBL2427005 0.86 MGLL (0.59) DRD2DRD1DRD4DRD5DRD3
SCHEMBL2348024 0.86 MGLL (0.56) GPR119MGLL
SCHEMBL29469965 0.83 MGLL (0.50) GPR119MGLL
SCHEMBL23867943 0.83 MGLL (0.50) GPR119MGLL
SCHEMBL23867878 0.83 MGLL (0.55) GPR119MGLL
SCHEMBL29470006 0.83 MGLL (0.55) GPR119MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2358704-A1 7-azaspiro [3.5]nonane-7-carboxamide compounds as modulators of fatty acid amide hydrolase Pfizer Inc. (US) 2011-08-24 EP disclosed
US-20100113465-A1 7-AZASPIRO[3.5]NONANE-7-CARBOXAMIDE COMPOUNDS PFIZER INC. 2010-05-06 US disclosed
WO-2010049841-A1 7-AZASPIRO [3.5] NONANE-7-CARBOXAMIDE COMPOUNDS AS MODULATORS OF FATTY ACID AMIDE HYDROLASE PFIZER INC. (US) 2010-05-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100113465-A1 7-AZASPIRO[3.5]NONANE-7-CARBOXAMIDE COMPOUNDS FAAH, FAAH2, APEH DRD2 1255/4885DRD1 1425/4885DRD4 2351/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.