SCHEMBL2349020

SCHEMBL2349020

CC(C)(C)NC(=O)Oc1c[nH]c2ncc(-c3cccc(N4CCCC4)c3)nc12

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SYK P43405 7/20 0.41
KCNH2 Q12809 1/20 0.41
MAP4K1 Q92918 3/20 0.40
PRKCI P41743 1/20 0.38
KIT P10721 1/20 0.38
WNT1 P04628 1/20 0.38
DYRK1A Q13627 1/20 0.38
MAPK1 P28482 1/20 0.38
CYP2D6 P10635 2/20 0.37
ATR Q13535 1/20 0.37
ROCK2 O75116 1/20 0.37
ROCK1 Q13464 1/20 0.37
JAK3 P52333 3/20 0.37
CYP2C9 P11712 1/20 0.36
ABL1 P00519 1/20 0.35
BCR P11274 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2344717 0.89 SYK (0.37) SYKKCNH2MAP4K1PRKCIMAPK1
SCHEMBL2342577 0.87 ALDH1A1 (0.40) SYKKCNH2MAPK1CYP2D6CYP2C9
SCHEMBL2362648 0.87 JAK3 (0.36) SYKKCNH2MAP4K1MAPK1CYP2D6
SCHEMBL2273872 0.84 SYK (0.58) SYKKCNH2CYP2D6
SCHEMBL2348276 0.81 SYK (0.38) SYKKCNH2MAP4K1PRKCICYP2D6
SCHEMBL2278709 0.80 JAK3 (0.55) SYKKCNH2PRKCIKITMAPK1
SCHEMBL2281125 0.79 JAK3 (0.54) SYKKCNH2PRKCIKITMAPK1
SCHEMBL2341691 0.78 SYK (0.43) SYKMAP4K1PRKCIJAK3CYP2C9
SCHEMBL2278520 0.78 JAK3 (0.55) SYKKCNH2PRKCIMAPK1CYP2D6
SCHEMBL2348404 0.78 SYK (0.55) SYKMAP4K1KITDYRK1AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245033-B1 PYRROLOPYRAZINE KINASE INHIBITORS HOFFMANN LA ROCHE (CH) 2011-08-31 EP claimed