SCHEMBL2362648

SCHEMBL2362648

COC1CCN(c2cccc(-c3cnc4[nH]cc(OC(=O)NC(C)(C)C)c4n3)c2)C1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 5/20 0.36
MAP4K1 Q92918 1/20 0.36
SYK P43405 3/20 0.35
IDH1 O75874 2/20 0.35
ADORA2A P29274 1/20 0.35
NEK2 P51955 1/20 0.34
CDC7 O00311 1/20 0.34
DBF4 Q9UBU7 1/20 0.34
LRRK2 Q5S007 2/20 0.34
KCNH2 Q12809 1/20 0.34
CYP2D6 P10635 1/20 0.34
TYRO3 Q06418 1/20 0.34
ATR Q13535 1/20 0.34
PDE2A O00408 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2275136 0.87 JAK3 (0.49) JAK3SYKKCNH2CYP2D6
SCHEMBL2349020 0.87 SYK (0.41) JAK3MAP4K1SYKKCNH2CYP2D6
SCHEMBL2349156 0.86 JAK3 (0.39) JAK3MAP4K1SYKADORA2A
SCHEMBL1892513 0.84 JAK3 (0.51) JAK3SYKIDH1ADORA2A
SCHEMBL2344717 0.83 SYK (0.37) JAK3MAP4K1SYKKCNH2CYP2D6
SCHEMBL3061667 0.82 PRKAB2 (0.43) JAK3MAP4K1SYKIDH1ADORA2A
SCHEMBL12372234 0.80 MAP4K1 (0.39) JAK3MAP4K1SYKIDH1ADORA2A
SCHEMBL2342577 0.80 ALDH1A1 (0.40) SYKKCNH2CYP2D6MAPK1
SCHEMBL3396539 0.78 JAK3 (0.36) JAK3MAP4K1IDH1ADORA2ACDC7
SCHEMBL2274966 0.76 JAK3 (0.52) JAK3SYKCYP2D6ATRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245033-B1 PYRROLOPYRAZINE KINASE INHIBITORS HOFFMANN LA ROCHE (CH) 2011-08-31 EP claimed