SCHEMBL23525828

SCHEMBL23525828

Cc1c(C#N)cccc1C(C)NC(=O)O

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 14/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
MAPK1 P28482 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CTSA P10619 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23525827 1.00 SOS1 (0.41) SOS1L3MBTL1MAPK1SMN1; SMN2CTSA
SCHEMBL30014414 1.00 SOS1 (0.41) SOS1L3MBTL1MAPK1SMN1; SMN2CTSA
SCHEMBL23525873 0.82 SOS1 (0.43) SOS1L3MBTL1MAPK1SMN1; SMN2CTSA
SCHEMBL30014661 0.82 SOS1 (0.43) SOS1L3MBTL1MAPK1SMN1; SMN2CTSA
SCHEMBL23525871 0.82 SOS1 (0.43) SOS1L3MBTL1MAPK1SMN1; SMN2CTSA
SCHEMBL28880409 0.82 TRPA1 (0.46)
SCHEMBL23563447 0.82 TRPA1 (0.46)
SCHEMBL29945842 0.82 TRPA1 (0.46)
SCHEMBL25628057 0.79 SOS1 (0.44) SOS1
SCHEMBL23526447 0.76 SOS1 (0.41) SOS1SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023250165-A1 SALTS OF SOS1 INHIBITORS Mirati Therapeutics, Inc. (US) 2023-12-28 WO disclosed
US-11702418-B2 SOS1 inhibitors Mirati Therapeutics, Inc. (US) 2023-07-18 US disclosed
US-20230137886-A1 SOS1 INHIBITORS Mirati Therapeutics, Inc. 2023-05-04 US disclosed
WO-2023030216-A1 QUINAZOLINE DERIVATIVE, OR PREPARATION METHOD THEREFOR AND USE THEREOF 浙江海正药业股份有限公司 2023-03-09 WO disclosed
US-20210188857-A1 SOS1 INHIBITORS Mirati Therapeutics, Inc. 2021-06-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230137886-A1 SOS1 INHIBITORS SOS1, SOS2, SAV1 SOS1 1/4885L3MBTL1 519/4885MAPK1 576/4885
US-20210188857-A1 SOS1 INHIBITORS SOS1, SOS2, SOST SOS1 1/4885L3MBTL1 1107/4885MAPK1 608/4885
US-11702418-B2 SOS1 inhibitors SOS1, SOS2, SOST SOS1 1/4885L3MBTL1 1107/4885MAPK1 608/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.