SCHEMBL2353237

SCHEMBL2353237

COC(=O)c1ccc(-c2cc(-c3ccc(C4CCCCC4)cc3)on2)cc1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 5/20 0.48
MAPT P10636 4/20 0.47
TP53 P04637 1/20 0.47
NPC1 O15118 6/20 0.45
RAB9A P51151 6/20 0.45
ALDH1A1 P00352 2/20 0.45
S1PR3 Q99500 1/20 0.44
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
SCD5 Q86SK9 2/20 0.44
SCD O00767 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
ABCB1 P08183 1/20 0.43
ABCC1 P33527 1/20 0.43
S1PR5 Q9H228 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12243237 0.88 S1PR1 (0.50) S1PR1MAPTNPC1RAB9AALDH1A1
SCHEMBL12243261 0.87 S1PR1 (0.56) S1PR1NPC1RAB9AS1PR3SCD5
SCHEMBL12243119 0.83 S1PR1 (0.45) S1PR1NPC1RAB9AS1PR3KMT2A
SCHEMBL15214831 0.82 ALDH1A1 (0.56) MAPTNPC1RAB9AALDH1A1KMT2A
SCHEMBL1790000 0.81 ALDH1A1 (0.59) MAPTNPC1RAB9AALDH1A1KMT2A
SCHEMBL2949436 0.81 ALDH1A1 (0.59) MAPTNPC1RAB9AALDH1A1KMT2A
SCHEMBL2944396 0.81 ALDH1A1 (0.59) MAPTNPC1RAB9AALDH1A1KMT2A
SCHEMBL5203862 0.80 NPC1 (0.65) MAPTTP53NPC1RAB9AALDH1A1
SCHEMBL12171876 0.80 RAB9A (0.61) MAPTTP53NPC1RAB9AALDH1A1
SCHEMBL5205950 0.80 NPC1 (0.65) MAPTTP53NPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8921309-B2 Lipopeptide compounds and their use UNIQUEST PTY LIMITED (AU) 2014-12-30 US disclosed
EP-2350119-B1 LIPOPEPTIDE COMPOUNDS AND THEIR USE UNIQUEST PTY LTD (AU) 2014-10-29 EP disclosed
EP-2350119-A1 LIPOPEPTIDE COMPOUNDS AND THEIR USE Merlion Pharmaceuticals Pte Ltd. (SG) 2011-08-03 EP disclosed
WO-2010062264-A1 LIPOPEPTIDE COMPOUNDS AND THEIR USE MERLION PHARMACEUTICALS PTE LTD (SG) 2010-06-03 WO disclosed