SCHEMBL23535233

SCHEMBL23535233

Nc1cc(Br)c(F)cc1CCO

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 8/20 0.38
KDM1B Q8NB78 5/20 0.38
KCNH2 Q12809 4/20 0.38
CA2 P00918 1/20 0.33
ADRB2 P07550 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31028666 0.84 KDM1A (0.36) KDM1AKDM1BKCNH2ADRB2CYP1A2
SCHEMBL31394862 0.78 KDM1A (0.32) KDM1AKDM1BKCNH2CA2CYP1A2
SCHEMBL31413426 0.76 TAAR1 (0.42) KDM1AKDM1BKCNH2
SCHEMBL17466051 0.76 KDM1A (0.32) KDM1AKDM1BKCNH2ADRB2CYP1A2
SCHEMBL30707419 0.76 KDM1A (0.32) KDM1AKDM1BKCNH2ADRB2CYP1A2
SCHEMBL3368244 0.75 CA2 (0.33) KDM1AKDM1BKCNH2CA2CYP1A2
SCHEMBL13310106 0.75 CYP1A2 (0.40) KDM1AKDM1BCYP1A2CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL31413389 0.74 TAAR1 (0.41) KDM1AKDM1BKCNH2
SCHEMBL31424538 0.74 CXCL8 (0.36) KDM1AKDM1BKCNH2
SCHEMBL30886492 0.74 KIF11 (0.34) KDM1AKDM1BKCNH2CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4076459-A1 PRMT5 INHIBITORS Merck Sharp & Dohme LLC (US) 2022-10-26 EP disclosed
WO-2021126728-A1 PRMT5 INHIBITORS MERCK SHARP & DOHME CORP. (US) 2021-06-24 WO disclosed