SCHEMBL23536251

SCHEMBL23536251

O=S(=O)(Cl)C=C(F)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.42
CYP2C19 P33261 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
MCOLN3 Q8TDD5 1/20 0.42
TDP1 Q9NUW8 3/20 0.38
HSD17B10 Q99714 2/20 0.38
CES1 P23141 4/20 0.36
CES2 O00748 3/20 0.36
TSHR P16473 3/20 0.36
DAO P14920 1/20 0.36
NAPRT Q6XQN6 1/20 0.36
MAPK1 P28482 2/20 0.35
AKR1C1 Q04828 2/20 0.35
MEN1 O00255 1/20 0.35
PABPC1 P11940 1/20 0.35
CCR6 P51684 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2024278 0.83 ALDH1A1 (0.45) ALDH1A1CYP2C19L3MBTL1CYP1A2CYP2C9
SCHEMBL29931991 0.79 ALDH1A1 (0.42) ALDH1A1CYP2C19L3MBTL1CYP1A2CYP2C9
SCHEMBL7372442 0.78 ALDH1A1 (0.61) ALDH1A1CYP2C19L3MBTL1CYP1A2CYP2C9
SCHEMBL11537148 0.75 ALDH1A1 (0.42) ALDH1A1CYP2C19L3MBTL1CYP1A2CYP2C9
SCHEMBL11537150 0.75 ALDH1A1 (0.42) ALDH1A1CYP2C19L3MBTL1CYP1A2CYP2C9
SCHEMBL3058443 0.75 ALDH1A1 (0.42) ALDH1A1CYP2C19L3MBTL1CYP1A2CYP2C9
SCHEMBL28122885 0.70 CES1 (0.38) ALDH1A1CYP2C19L3MBTL1TDP1HSD17B10
SCHEMBL8562028 0.69 ALDH1A1 (0.55) ALDH1A1CYP2C19L3MBTL1CYP1A2CYP2C9
SCHEMBL6832826 0.68 NFE2L2 (0.43) ALDH1A1CYP2C19L3MBTL1TDP1HSD17B10
SCHEMBL4135542 0.68 ALDH1A1 (0.38) ALDH1A1CYP2C19L3MBTL1CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4076423-A1 TRPML MODULATORS Casma Therapeutics, Inc. (US) 2022-10-26 EP disclosed
WO-2021127337-A1 TRPML MODULATORS CASMA THERAPEUTICS, INC. (US) 2021-06-24 WO disclosed