SCHEMBL23536396

SCHEMBL23536396

Nc1ccccc1C1=CCN(c2ccc(Cl)cc2F)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
LMNA P02545 2/20 0.39
KDM4E B2RXH2 1/20 0.39
HTT P42858 1/20 0.39
DRD4 P21917 1/20 0.39
GRM2 Q14416 1/20 0.39
OPRM1 P35372 1/20 0.37
OPRK1 P41145 1/20 0.37
MAPT P10636 1/20 0.36
MAPK1 P28482 1/20 0.36
GFER P55789 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
HTR1A P08908 1/20 0.36
POLB P06746 1/20 0.35
TRPV1 Q8NER1 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A3 Q01959 1/20 0.35
SMARCA2 P51531 1/20 0.34
DRD2 P14416 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29932060 1.00 ALDH1A1 (0.39) ALDH1A1LMNAKDM4EHTTDRD4
SCHEMBL29931935 0.81 ALDH1A1 (0.44) ALDH1A1LMNAHTTMAPTMAPK1
SCHEMBL23536527 0.81 ALDH1A1 (0.44) ALDH1A1LMNAHTTMAPTMAPK1
SCHEMBL21261239 0.74 POLB (0.54) ALDH1A1LMNAKDM4EHTTDRD4
SCHEMBL29931958 0.74 DRD4 (0.38) ALDH1A1DRD4GRM2POLBTRPV1
SCHEMBL23536237 0.74 DRD4 (0.38) ALDH1A1DRD4GRM2POLBTRPV1
SCHEMBL29931990 0.72 DRD4 (0.39) ALDH1A1LMNADRD4GRM2MAPT
SCHEMBL23536130 0.70 ALDH1A1 (0.42) ALDH1A1LMNAKDM4EHTTDRD4
SCHEMBL29932056 0.70 ALDH1A1 (0.42) ALDH1A1LMNAKDM4EHTTDRD4
SCHEMBL24628435 0.68 ALDH1A1 (0.41) ALDH1A1LMNAKDM4EHTTDRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4076423-A1 TRPML MODULATORS Casma Therapeutics, Inc. (US) 2022-10-26 EP disclosed
WO-2021127337-A1 TRPML MODULATORS CASMA THERAPEUTICS, INC. (US) 2021-06-24 WO disclosed