SCHEMBL23536504

SCHEMBL23536504

Cn1nc(C2CCN(c3ccc(Cl)cc3F)CC2)nc1N

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 1/20 0.42
GRM2 Q14416 1/20 0.42
POLB P06746 1/20 0.39
PHGDH O43175 1/20 0.39
ADORA2A P29274 3/20 0.38
HTR3A P46098 1/20 0.37
HRH4 Q9H3N8 1/20 0.37
ALDH1A1 P00352 2/20 0.36
HTT P42858 2/20 0.36
ADORA2B P29275 1/20 0.35
DPP4 P27487 1/20 0.35
DPP8 Q6V1X1 1/20 0.35
DPP9 Q86TI2 1/20 0.35
DPP7 Q9UHL4 1/20 0.35
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35
TRPA1 O75762 1/20 0.35
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
HTR1A P08908 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29931890 1.00 DRD4 (0.42) DRD4GRM2POLBPHGDHADORA2A
SCHEMBL23536434 0.81 DRD4 (0.47) DRD4GRM2POLBPHGDHADORA2A
SCHEMBL29931887 0.81 DRD4 (0.47) DRD4GRM2POLBPHGDHADORA2A
SCHEMBL23536198 0.79 GRM2 (0.40) DRD4GRM2POLBPHGDHADORA2A
SCHEMBL23536212 0.75 HRH4 (0.47) POLBHRH4ALDH1A1LMNA
SCHEMBL29931770 0.73 DRD4 (0.47) DRD4GRM2POLBPHGDHADORA2A
SCHEMBL23536253 0.73 DRD4 (0.47) DRD4GRM2POLBPHGDHADORA2A
SCHEMBL29931979 0.72 SSTR2 (0.45) DRD4GRM2POLBPHGDHHTR3A
SCHEMBL23536333 0.72 SSTR2 (0.45) DRD4GRM2POLBPHGDHHTR3A
SCHEMBL30232382 0.72 GRM2 (0.42) DRD4GRM2POLBPHGDHDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115087440-A TRPML modulators 卡斯玛治疗公司 2022-09-20 CN disclosed
WO-2021127337-A1 TRPML MODULATORS CASMA THERAPEUTICS, INC. (US) 2021-06-24 WO disclosed